Compile Data Set for Download or QSAR
Report error Found 73 Enz. Inhib. hit(s) with all data for entry = 5399
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86123(LDHA Inhibitor, 18)
Affinity DataKd:  1.70E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86136(LDHA Inhibitor, 32)
Affinity DataKd:  180nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86135(LDHA Inhibitor, 31)
Affinity DataKd:  60nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataKd:  1.20E+3nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86133(LDHA Inhibitor, 29)
Affinity DataKd:  69nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86132(LDHA Inhibitor, 28)
Affinity DataKd:  3.20E+3nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86120(LDHA Inhibitor, 15)
Affinity DataKd:  7.90E+5nMpH: 7.5Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86121(LDHA Inhibitor, 16)
Affinity DataKd:  5.00E+5nMpH: 7.5Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86122(LDHA Inhibitor, 17)
Affinity DataKd:  4.00E+4nMpH: 7.5Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86123(LDHA Inhibitor, 18)
Affinity DataKd:  1.30E+5nMpH: 7.5Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86121(LDHA Inhibitor, 16)
Affinity DataKd:  5.40E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86122(LDHA Inhibitor, 17)
Affinity DataKd:  9.20E+4nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataKd:  93nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86131(LDHA Inhibitor, 27)
Affinity DataKd:  46nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataKd:  130nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86129(LDHA Inhibitor, 25)
Affinity DataKd:  2.40E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86129(LDHA Inhibitor, 25)
Affinity DataKd:  1.10E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataKd:  2.10E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86125(LDHA Inhibitor, 21)
Affinity DataKd:  2.80E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86124(LDHA Inhibitor, 20)
Affinity DataKd:  4.70E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86125(LDHA Inhibitor, 21)
Affinity DataKd:  1.00E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86128(LDHA Inhibitor, 24)
Affinity DataKd:  1.60E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86127(LDHA Inhibitor, 23)
Affinity DataKd:  3.50E+4nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86126(LDHA Inhibitor, 22)
Affinity DataKd:  7.70E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86117(LDHA Inhibitor, 12)
Affinity DataKd:  7.70E+5nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86138(LDHA Inhibitor, 34)
Affinity DataKd:  8nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Astrazeneca

LigandPNGBDBM86114(LDHA Inhibitor, 8)
Affinity DataKd:  1.28E+4nMpH: 7.4 T: 2°CAssay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Astrazeneca

LigandPNGBDBM50339607(LDHA Inhibitor, 4 | CHEMBL1688790 | 1-Hydroxy-6-ph...)
Affinity DataKd:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Astrazeneca

LigandPNGBDBM50219487(CHEMBL229299 | LDHA Inhibitor, 5 | 1-hydroxy-2-nap...)
Affinity DataKd:  6.40E+5nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Astrazeneca

LigandPNGBDBM50192453([(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihyd...)
Affinity DataKd:  6.50E+5nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Human)
Astrazeneca

LigandPNGBDBM86113(LDHA Inhibitor, 7)
Affinity DataKd:  4.00E+6nMpH: 7.5 T: 2°CAssay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86115(LDHA Inhibitor, 9)
Affinity DataKd:  3.00E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM50078827(CHEMBL83103 | LDHA Inhibitor, 10 | 2-Pyridin-3-yl-...)
Affinity DataKd:  1.40E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86116(LDHA Inhibitor, 11)
Affinity DataKd:  2.40E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86117(LDHA Inhibitor, 12)
Affinity DataKd:  1.00E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86118(LDHA Inhibitor, 13)
Affinity DataKd:  4.00E+5nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86119(LDHA Inhibitor, 14)
Affinity DataKd:  4.20E+6nMpH: 7.5Assay Description:NMR spectra were acquired on Bruker Avance 600 MHz spectrometers at 298 K using a 5 mm triple-resonance HCN cryoprobe. Ligand binding was detected u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86115(LDHA Inhibitor, 9)
Affinity DataKd:  1.60E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86116(LDHA Inhibitor, 11)
Affinity DataKd:  3.00E+6nMpH: 7.4Assay Description:A BIAcore 3000 or a BIAcore S51 instrument (GE Healthcare) was used to detect binding interactions using a direct binding assay format.More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86138(LDHA Inhibitor, 34)
Affinity DataIC50: 270nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86135(LDHA Inhibitor, 31)
Affinity DataIC50: 290nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86137(LDHA Inhibitor, 33)
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86133(LDHA Inhibitor, 29)
Affinity DataIC50: 1.90E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86131(LDHA Inhibitor, 27)
Affinity DataIC50: 3.10E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86130(LDHA Inhibitor, 26)
Affinity DataIC50: 4.20E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86136(LDHA Inhibitor, 32)
Affinity DataIC50: 7.40E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Human)
Astrazeneca

LigandPNGBDBM23251(4-hydroxy-1,2,5-thiadiazole-3-carboxylic acid | LD...)
Affinity DataIC50: 7.80E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase B chain(Human)
Astrazeneca

LigandPNGBDBM86114(LDHA Inhibitor, 8)
Affinity DataIC50: 9.40E+3nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86134(LDHA Inhibitor, 30)
Affinity DataIC50: 2.95E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
TargetL-lactate dehydrogenase A chain(Rat)
Astrazeneca

LigandPNGBDBM86132(LDHA Inhibitor, 28)
Affinity DataIC50: 8.62E+4nMpH: 7.5 T: 2°CAssay Description:Enzyme assay using lactate dehydrogenase A (LDHA).More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/21/2012
Entry Details Article
PubMed
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