Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 8319
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240828((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
Affinity DataIC50: 1.26E+3nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 2.55E+3nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240829((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 4.40E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240824((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 5.67E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240824((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 6.46E+4nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240825((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 7.70E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240827((2S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanam...)
Affinity DataIC50: 8.29E+4nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240823((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 1.05E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240825((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 1.28E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240831((2R,3S)-3-amino-2-hydroxy-N-((S)-3-hydroxy-1-(hydr...)
Affinity DataIC50: 1.58E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM23971(CHEMBL29292 | (2S)-2-[(2S,3R)-3-amino-2-hydroxy-4-...)
Affinity DataIC50: 1.63E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240830((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 1.73E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240822((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 1.86E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240816((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 1.98E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240827((2S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanam...)
Affinity DataIC50: 2.07E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240828((2R,3S)-3-amino-2-hydroxy-N-((S)-2-(hydroxyamino)-...)
Affinity DataIC50: 2.13E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240812((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 2.15E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240829((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 2.49E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240816((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 2.54E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240815((2S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanam...)
Affinity DataIC50: 2.64E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240814((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 2.73E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240813((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 2.87E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240826((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 2.92E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240831((2R,3S)-3-amino-2-hydroxy-N-((S)-3-hydroxy-1-(hydr...)
Affinity DataIC50: 2.92E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240830((2R,3S)-3-amino-2-hydroxy-N-((S)-1-(hydroxyamino)-...)
Affinity DataIC50: 2.99E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240814((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.42E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240812((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.52E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240832((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 3.63E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240818((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 4.07E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240821((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 4.24E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240817((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 4.97E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240821((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 5.13E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240819((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpropanami...)
Affinity DataIC50: 5.62E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
TargetAminopeptidase N(Pig)
Shandong University

LigandPNGBDBM240820((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 5.90E+5nMpH: 7.5 T: 2°CAssay Description:IC50 values against APN from Porcine Kidney were determined by using L-Leu-p-nitroanilide as a substrate. All the solutions of the inhibitors were pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Pig)
Shandong University

LigandPNGBDBM240820((S)-2-((S)-2-((2R,3S)-3-amino-2-hydroxy-3-phenylpr...)
Affinity DataIC50: 6.90E+5nMAssay Description:Gelatinase A (MMP-2) and TNBS were purchased from Sigma, and the substance was synthesized as described by Vijaykumar et al. The gelatinase, substanc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2017
Entry Details Article
PubMed