Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50034644
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365592(CHEMBL1957805)
Affinity DataKi:  0.400nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365589(CHEMBL1957802)
Affinity DataKi:  0.600nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365586(CHEMBL1957801)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50324551((4-Bromo-1-methyl-1H-pyrazol-3-yl)-{4-[2-(2,4-difl...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365595(CHEMBL1957812)
Affinity DataKi:  1.40nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365590(CHEMBL1957818)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365581(CHEMBL1957817)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365579(CHEMBL1957814)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365591(CHEMBL1957803)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365583(CHEMBL1957811)
Affinity DataKi:  1.90nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365580(CHEMBL1957808)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365593(CHEMBL1957813)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365574(CHEMBL1957819)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365577(CHEMBL1957815)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365594(CHEMBL1957821)
Affinity DataKi:  3.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365578(CHEMBL1957807)
Affinity DataKi:  3.80nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365582(CHEMBL1957810)
Affinity DataKi:  4.30nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365587(CHEMBL1957820)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365576(CHEMBL1957806)
Affinity DataKi:  5.60nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365588(CHEMBL1957800)
Affinity DataKi:  5.70nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365584(CHEMBL1957804)
Affinity DataKi:  5.90nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365575(CHEMBL1957809)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365595(CHEMBL1957812)
Affinity DataKi:  152nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365594(CHEMBL1957821)
Affinity DataKi:  153nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365593(CHEMBL1957813)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365592(CHEMBL1957805)
Affinity DataKi:  194nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365591(CHEMBL1957803)
Affinity DataKi:  246nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365590(CHEMBL1957818)
Affinity DataKi:  391nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365589(CHEMBL1957802)
Affinity DataKi:  394nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365588(CHEMBL1957800)
Affinity DataKi:  467nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365587(CHEMBL1957820)
Affinity DataKi:  474nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365586(CHEMBL1957801)
Affinity DataKi:  496nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataKi:  524nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365584(CHEMBL1957804)
Affinity DataKi:  575nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365583(CHEMBL1957811)
Affinity DataKi:  581nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365582(CHEMBL1957810)
Affinity DataKi:  596nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365581(CHEMBL1957817)
Affinity DataKi:  682nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365580(CHEMBL1957808)
Affinity DataKi:  717nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365579(CHEMBL1957814)
Affinity DataKi:  739nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365578(CHEMBL1957807)
Affinity DataKi:  910nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365577(CHEMBL1957815)
Affinity DataKi:  997nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365576(CHEMBL1957806)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human ERG by patch-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50324551((4-Bromo-1-methyl-1H-pyrazol-3-yl)-{4-[2-(2,4-difl...)
Affinity DataKi:  2.82E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365575(CHEMBL1957809)
Affinity DataKi:  2.88E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365574(CHEMBL1957819)
Affinity DataKi:  6.90E+3nMAssay Description:Displacement of [125I]-DOI from recombinant human 5HT2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP2D6 in human liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP219 in human liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50365585(CHEMBL1957816)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
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