Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50004608
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50484729(CHEMBL1949982)
Affinity DataEC50:  1.40E+3nMAssay Description:Corrector activity at human CFTR delta F508 mutant expressed in rat FRT cells coexpressing fluorescent protein YFP-H148Q/1152L by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50484730(CHEMBL1949981)
Affinity DataEC50:  1.40E+3nMAssay Description:Corrector activity at human CFTR delta F508 mutant expressed in rat FRT cells coexpressing fluorescent protein YFP-H148Q/1152L by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed
TargetCystic fibrosis transmembrane conductance regulator(Human)
University of California Davis

Curated by ChEMBL
LigandPNGBDBM50289704(CHEMBL260775)
Affinity DataEC50:  2.30E+3nMAssay Description:Corrector activity at human CFTR delta F508 mutant expressed in rat FRT cells coexpressing fluorescent protein YFP-H148Q/1152L by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2020
Entry Details Article
PubMed