Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50034582
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sanofi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364664(CHEMBL1951453)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ERG by whole-cell patch clamp electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Sanofi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364664(CHEMBL1951453)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human CYP2D6 using dexotromethorphan as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364664(CHEMBL1951453)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human CYP3A4 using midazolam as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Sanofi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364665(CHEMBL1951454)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human CYP3A4 using midazolam as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Sanofi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50364665(CHEMBL1951454)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of human CYP2D6 using dexotromethorphan as substrate by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed