Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50034574
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364466(CHEMBL1950695)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364465(CHEMBL1950694)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364465(CHEMBL1950694)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364468(CHEMBL1950698)
Affinity DataIC50: 41nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364464(CHEMBL1950693)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364469(CHEMBL1950696)
Affinity DataIC50: 46nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364468(CHEMBL1950698)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364467(CHEMBL1950697)
Affinity DataIC50: 61nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364466(CHEMBL1950695)
Affinity DataIC50: 65nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364467(CHEMBL1950697)
Affinity DataIC50: 85nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364464(CHEMBL1950693)
Affinity DataIC50: 101nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activity after 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetGlucocorticoid receptor(Human)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50364469(CHEMBL1950696)
Affinity DataIC50: 142nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of dexamethasone-induced transcription at GRE after 24 hrs ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed