Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50004775
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50173647(4-[(E)-2-(4-Methylamino-phenyl)-vinyl]-phenol | [3...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to amyloid beta (1-42) aggregates in human Alzheimer's disease brain sectionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50485236(CHEBI:79033 | BAY-949172 | Florbetaben (18f) | Flo...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to amyloid beta (1-42) aggregates in human Alzheimer's disease brain sectionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Sungkyunkwan University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50484946(CHEBI:66880 | (18F)AV-45 | 18F-AV-45 | AV-45 F-18 ...)
Affinity DataKi:  2.90nMAssay Description:Binding affinity to amyloid beta (1-42) aggregates in human Alzheimer's disease brain sectionsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed