Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50034375
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50100436(CHEMBL412768 | NH2-Lys-Thr-Glu-Glu-Ile-Ser-Glu-Val...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361388(CHEMBL1934195)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361391(CHEMBL1934197)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361381(CHEMBL1412710)
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50310823(bergamottin | CHEMBL1078442)
Affinity DataIC50: 3.22E+4nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50308719(Imperatorin | (9-[(3-methyl-2-buten-1-yl)oxy]-7H-f...)
Affinity DataIC50: 9.18E+4nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361389(CHEMBL1934196)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361390(BYAKANGELICIN)
Affinity DataIC50: 2.20E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50242377(isoimperatorin | CHEMBL448060)
Affinity DataIC50: 2.44E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361373(AURAPTENE)
Affinity DataIC50: 3.45E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361376(OXYPEUCEDANIN)
Affinity DataIC50: 3.59E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50292574(7-demethylsuberosine | CHEMBL502689)
Affinity DataIC50: 4.13E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361379(HERACLENIN)
Affinity DataIC50: 4.44E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50240868(CHEMBL350475 | 7-Hydroxy-8-(3-methyl-but-2-enyl)-c...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361385(CHEMBL1934071)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361377(CHEMBL454060)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50250917((2S)-2-(1-hydroxy-1-methylethyl)-2,3-dihydro-7H-fu...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50303499(7-(methyloxy)-2H-chromen-2-one | 7-Methoxycoumarin...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50067880(4-methoxy-7H-furo[3,2-g]chromen-7-one | 5-methoxyp...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361384(CHEMBL1934070)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361394(CHEMBL1934198)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361382(CHEMBL1934068)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361383(CHEMBL1934069)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361380(HERACLENOL)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50331545(2H-furo[2,3-h]chromen-2-one | Furo[2,3-h]chromen-2...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50331544(7H-furo[3,2-g]chromen-7-one | Furo[3,2-g]chromen-7...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50174558(umbelliferone | CHEMBL51628 | skimmetin | Coumarin...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50240512(osthole | 7-Methoxy-8-(3-methyl-but-2-enyl)-chrome...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361393(COLUMBIANETIN)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361398(CHEMBL503137 | LOMATIN)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361378(XANTHOTOXOL)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361397(CHEMBL71358)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM34571(6,7-dihydroxychromen-2-one | 6,7-dihydroxy-1-benzo...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361386(ISOPIMPINELLIN)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361372(CHEMBL156692)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361396((S)-(+)-Decursin | DECURSIN)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50259817(decursinol | CHEMBL481657)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50209569(4-hydroxy-7H-furo[3,2-g]chromen-7-one | bergaptol ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50041234(9-methoxy-7H-furo[3,2-g]chromen-7-one | CHEMBL416 ...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361375(CHEMBL1928409)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361392(CHEMBL1710181)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361395(CHEMBL1631595)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50292575(8,8-Dimethyl-8H-pyrano[3,2-g]chromen-2-one | CHEMB...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM12342(2H-chromen-2-one | CHEMBL6466 | Coumarin)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361374(SCOPARONE)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM81058(MLS000574895 | cid_98608 | SMR000156210 | 4-methox...)
Affinity DataIC50: 1.43E+6nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361387(CHEMBL1934194)
Affinity DataIC50: 3.44E+6nMAssay Description:Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50310823(bergamottin | CHEMBL1078442)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant human BACE1 assessed as dissociation constant of enzyme-substrate-inhibitor complex using Rh-EVNLDAEFK as substrate by Dixo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361390(BYAKANGELICIN)
Affinity DataKi:  6.20E+3nMAssay Description:Inhibition of recombinant human BACE1 assessed as dissociation constant of enzyme-substrate-inhibitor complex using Rh-EVNLDAEFK as substrate by Dixo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetBeta-secretase 1(Human)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50361388(CHEMBL1934195)
Affinity DataKi:  1.37E+4nMAssay Description:Inhibition of recombinant human BACE1 assessed as dissociation constant of enzyme-substrate-inhibitor complex using Rh-EVNLDAEFK as substrate by Dixo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
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