Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50006065
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496699(CHEMBL3220716)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496700(CHEMBL3220717)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496700(CHEMBL3220717)
Affinity DataKd:  1.80E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496701(CHEMBL3220718)
Affinity DataKd:  1.80E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496701(CHEMBL3220718)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed
TargetVitamin D3 receptor A(Zebrafish)
Centre National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50496699(CHEMBL3220716)
Affinity DataKd:  3.30E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2020
Entry Details Article
PubMed