Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50034289
TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360001(CHEMBL1928322)
Affinity DataEC50:  1.74E+4nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360002(CHEMBL1928323)
Affinity DataEC50:  1.66E+4nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50029051(4-[(1R)-2-amino-1-hydroxyethyl]benzene-1,2-diol | ...)
Affinity DataEC50:  118nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360000(CHEMBL1928316)
Affinity DataEC50:  4.50E+3nMAssay Description:Agonist activity at human adrenoceptor alpha2A expressed in CHOK1 cells assessed as stimulation of agonist-induced [35S]GTPgammaS binding by scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360020(CHEMBL1928335)
Affinity DataIC50: 646nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360002(CHEMBL1928323)
Affinity DataIC50: 856nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360005(CHEMBL1928319)
Affinity DataIC50: 5.15E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360010(CHEMBL1928326)
Affinity DataIC50: 9.39E+3nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360004(CHEMBL1928318)
Affinity DataIC50: 1.29E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360008(CHEMBL1928324)
Affinity DataIC50: 1.64E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360018(CHEMBL1928334)
Affinity DataIC50: 1.68E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360000(CHEMBL1928316)
Affinity DataIC50: 1.94E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360013(CHEMBL1928329)
Affinity DataIC50: 2.10E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360003(CHEMBL1928317)
Affinity DataIC50: 2.13E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360012(CHEMBL1928328)
Affinity DataIC50: 2.81E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360006(CHEMBL1928320)
Affinity DataIC50: 3.29E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360009(CHEMBL1928325)
Affinity DataIC50: 4.39E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360011(CHEMBL1928327)
Affinity DataIC50: 4.42E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360007(CHEMBL1928321)
Affinity DataIC50: 4.54E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360019(CHEMBL1926702)
Affinity DataIC50: 4.88E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360017(CHEMBL1928333)
Affinity DataIC50: 5.68E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360015(CHEMBL1928331)
Affinity DataIC50: 7.40E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360014(CHEMBL1928330)
Affinity DataIC50: 7.77E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360016(CHEMBL1928332)
Affinity DataIC50: 9.33E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNischarin(Rat)
Medical University of Gdansk

Curated by ChEMBL
LigandPNGBDBM50360001(CHEMBL1928322)
Affinity DataIC50: 9.64E+4nMAssay Description:Displacement of [3H]clonidine from imidazoline I1 receptor in Sprague-Dawley rat kidney membranes after 45 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed