Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50034473
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363052BDBM50363052(CHEMBL1946956)
Affinity DataEC50:  60nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343350BDBM50343350(4,4,4-trifluoro-1-(4-(3-(thiophen-2-yl)-1,2,4-oxad...)
Affinity DataEC50:  100nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363017BDBM50363017(CHEMBL1945812)
Affinity DataEC50:  200nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343351BDBM50343351(4,4,4-Trifluoro-1-[(R)-3-(3-thiophen-2-yl-1,2,4-ox...)
Affinity DataEC50:  400nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363052BDBM50363052(CHEMBL1946956)
Affinity DataIC50: 400nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363015BDBM50363015(CHEMBL1945701)
Affinity DataEC50:  500nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363018BDBM50363018(CHEMBL1945813)
Affinity DataEC50:  500nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363044BDBM50363044(CHEMBL1946419)
Affinity DataEC50:  800nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363042BDBM50363042(CHEMBL1946417)
Affinity DataEC50:  800nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363045BDBM50363045(CHEMBL1946420)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363017BDBM50363017(CHEMBL1945812)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363025BDBM50363025(CHEMBL1945820)
Affinity DataEC50:  1.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363029BDBM50363029(CHEMBL1945962)
Affinity DataEC50:  1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363030BDBM50363030(CHEMBL1945963)
Affinity DataEC50:  1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363014BDBM50363014(CHEMBL1945700)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343350BDBM50343350(4,4,4-trifluoro-1-(4-(3-(thiophen-2-yl)-1,2,4-oxad...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50343351BDBM50343351(4,4,4-Trifluoro-1-[(R)-3-(3-thiophen-2-yl-1,2,4-ox...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363032BDBM50363032(CHEMBL1945965)
Affinity DataEC50:  2.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363031BDBM50363031(CHEMBL1945964)
Affinity DataEC50:  2.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363016BDBM50363016(CHEMBL1945811)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363038BDBM50363038(CHEMBL1945971)
Affinity DataEC50:  2.50E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363015BDBM50363015(CHEMBL1945701)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363047BDBM50363047(CHEMBL1946422)
Affinity DataEC50:  3.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363049BDBM50363049(CHEMBL1946424)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363043BDBM50363043(CHEMBL1946418)
Affinity DataEC50:  4.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363022BDBM50363022(CHEMBL1945817)
Affinity DataEC50:  4.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363048BDBM50363048(CHEMBL1946423)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363050BDBM50363050(CHEMBL1946425)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363046BDBM50363046(CHEMBL1946421)
Affinity DataEC50: >5.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363027BDBM50363027(CHEMBL1945821)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363051BDBM50363051(CHEMBL1946426)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363026BDBM50363026(CHEMBL1944650)
Affinity DataEC50:  7.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363020BDBM50363020(CHEMBL1945815)
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363018BDBM50363018(CHEMBL1945813)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of EthR binding to ethA promoter in 106-bp biotinylated DNA preincubated for 5 mins measured for 3 mins by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363023BDBM50363023(CHEMBL1945818)
Affinity DataEC50:  9.30E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363034BDBM50363034(CHEMBL1945967)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363033BDBM50363033(CHEMBL1945966)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363028BDBM50363028(CHEMBL1945961)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363024BDBM50363024(CHEMBL1945819)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363040BDBM50363040(CHEMBL1946415)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363039BDBM50363039(CHEMBL1945972)
Affinity DataEC50:  1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363041BDBM50363041(CHEMBL1946416)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363036BDBM50363036(CHEMBL1945969)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363035BDBM50363035(CHEMBL1945968)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363021BDBM50363021(CHEMBL1945816)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363037BDBM50363037(CHEMBL1945970)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetHTH-type transcriptional regulator EthR(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Lille

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363019BDBM50363019(CHEMBL1945814)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis H37Rv EthR in Mycobacterium tuberculosis H37Rv expressing GFP infected mouse in RAW264.7 cells assessed as p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed