Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50034472
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363009BDBM50363009(CHEMBL1946412)
Affinity DataIC50: 200nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363013BDBM50363013(CHEMBL191539)
Affinity DataIC50: 240nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363006BDBM50363006(CHEMBL363989)
Affinity DataIC50: 280nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363004BDBM50363004(CHEMBL1946140)
Affinity DataIC50: 350nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130735BDBM50130735((7-chloro-1,1-dioxo-1,4-dihydro-benzo[1,2,4]thiadi...)
Affinity DataIC50: 480nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363007BDBM50363007(CHEMBL1946272)
Affinity DataIC50: 520nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362998BDBM50362998(CHEMBL1945810)
Affinity DataIC50: 620nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363002BDBM50363002(CHEMBL115565)
Affinity DataIC50: 760nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363003BDBM50363003(CHEMBL1946139)
Affinity DataIC50: 1.41E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363008BDBM50363008(CHEMBL1946410)
Affinity DataIC50: 1.67E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362992BDBM50362992(CHEMBL1946411)
Affinity DataIC50: 1.73E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363011BDBM50363011(CHEMBL189093)
Affinity DataIC50: 1.75E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362991BDBM50362991(CHEMBL1946273)
Affinity DataIC50: 1.81E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363001BDBM50363001(CHEMBL1946137)
Affinity DataIC50: 2.05E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363012BDBM50363012(CHEMBL1946759)
Affinity DataIC50: 2.98E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362995BDBM50362995(CHEMBL1945807)
Affinity DataIC50: 3.03E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362997BDBM50362997(CHEMBL1945809)
Affinity DataIC50: 3.58E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362990BDBM50362990(CHEMBL1946138)
Affinity DataIC50: 3.78E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363010BDBM50363010(CHEMBL1946414)
Affinity DataIC50: 4.93E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362993BDBM50362993(CHEMBL1944656)
Affinity DataIC50: 6.31E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363005BDBM50363005(CHEMBL1946270)
Affinity DataIC50: 8.67E+3nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362990BDBM50362990(CHEMBL1946138)
Affinity DataIC50: 1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362992BDBM50362992(CHEMBL1946411)
Affinity DataIC50: 1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362991BDBM50362991(CHEMBL1946273)
Affinity DataIC50: 1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362994BDBM50362994(CHEMBL1946760)
Affinity DataIC50: 1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362993BDBM50362993(CHEMBL1944656)
Affinity DataIC50: 1.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50363000BDBM50363000(CHEMBL1946136)
Affinity DataIC50: 2.65E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362999BDBM50362999(CHEMBL1946134)
Affinity DataIC50: 3.75E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362996BDBM50362996(CHEMBL1945808)
Affinity DataIC50: 3.89E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetATP-binding cassette sub-family C member 8(Rat)
University of Liege

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50362989BDBM50362989(CHEMBL1945806)
Affinity DataIC50: 5.00E+4nMAssay Description:Activation of SUR1 in rat pancreatic islets assessed as inhibition of glucose-induced insulin secretionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed