Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50034082
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356624(CHEMBL1910278)
Affinity DataIC50: 90nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356616(CHEMBL1910270)
Affinity DataIC50: 300nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356618(CHEMBL1910272)
Affinity DataIC50: 500nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356622(CHEMBL1910276)
Affinity DataIC50: 900nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356623(CHEMBL1910277)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356621(CHEMBL1910275)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356620(CHEMBL1910274)
Affinity DataIC50: 6.30E+3nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM5718(2,6,9-Trisubstituted purine deriv. 26 | 2-{[6-(ben...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356625(CHEMBL1910279)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356617(CHEMBL1910271)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356615(CHEMBL1910269)
Affinity DataIC50: 2.95E+4nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356619(CHEMBL1910273)
Affinity DataIC50: 2.95E+4nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356614(CHEMBL1910268)
Affinity DataIC50: 2.95E+4nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356619(CHEMBL1910273)
Affinity DataIC50: 3.63E+4nMAssay Description:Inhibition of CDK2/cyclin A expressed in baculovirus infected insect Sf21 cells using [gamma-P32]ATP and histone H1 as substrate after 10 mins by rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356621(CHEMBL1910275)
Affinity DataIC50: 4.79E+4nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356624(CHEMBL1910278)
Affinity DataIC50: 6.61E+4nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356614(CHEMBL1910268)
Affinity DataIC50: 9.33E+4nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356615(CHEMBL1910269)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356616(CHEMBL1910270)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356617(CHEMBL1910271)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356618(CHEMBL1910272)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356620(CHEMBL1910274)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356622(CHEMBL1910276)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356623(CHEMBL1910277)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
National Organization For Drug Control & Research

Curated by ChEMBL
LigandPNGBDBM50356625(CHEMBL1910279)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed