Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50034054
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
Max Planck Research Unit For Enzymology of Protein Folding

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKd:  7.60nMAssay Description:Binding affinity to human recombinant cyclophilin-A by isothermal titration calorimetry assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
Max Planck Research Unit For Enzymology of Protein Folding

Curated by ChEMBL
LigandPNGBDBM50356016(CHEMBL1911379)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of PPIase activity of human recombinant cyclophilin-A using succinyl-Ala-Ala-Pro-Phe-4-nitroanilide as substrate by protease coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
Max Planck Research Unit For Enzymology of Protein Folding

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of PPIase activity of human recombinant cyclophilin-A using succinyl-Ala-Ala-Pro-Phe-4-nitroanilide as substrate by protease coupled assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed