Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50033926
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50168789(3-[1-(4-Chloro-benzyl)-3-methyl-1H-indol-2-yl]-2,2...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of microsomal PGESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50168789(3-[1-(4-Chloro-benzyl)-3-methyl-1H-indol-2-yl]-2,2...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human recombinant microsomal PGES-1 expressed in freestyle 293-f cells assessed as conversion of PGH2 to PGE2 after 15 mins by enzyme i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50353950(CHEMBL1828850)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of human recombinant microsomal PGES-1 expressed in freestyle 293-f cells assessed as conversion of PGH2 to PGE2 after 15 mins by enzyme i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50353951(CHEMBL1828851)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of human recombinant microsomal PGES-1 expressed in freestyle 293-f cells assessed as conversion of PGH2 to PGE2 after 15 mins by enzyme i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | NS398 | NS-398 | N-(2-Cyclohexyloxy-4...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of microsomal PGESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetProstaglandin E synthase(Human)
University of Kentucky

Curated by ChEMBL
LigandPNGBDBM50012899(cis-5-Fluoro-2-methyl-1-((p-methylsulfinyl)benzyli...)
Affinity DataIC50: 8.00E+4nMAssay Description:Inhibition of microsomal PGESMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed