Compile Data Set for Download or QSAR
Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50033994
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355111(CHEMBL1835210)
Affinity DataIC50: 12nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355109(CHEMBL1835209)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355101(CHEMBL1835324)
Affinity DataIC50: 22nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355099(CHEMBL1835322)
Affinity DataIC50: 24nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355099(CHEMBL1835322)
Affinity DataIC50: 26nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355110(CHEMBL1835208)
Affinity DataIC50: 29nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355110(CHEMBL1835208)
Affinity DataIC50: 41nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355111(CHEMBL1835210)
Affinity DataIC50: 41nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355109(CHEMBL1835209)
Affinity DataIC50: 46nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355103(CHEMBL1835399)
Affinity DataIC50: 50nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355094(CHEMBL1835317)
Affinity DataIC50: 50nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355112(CHEMBL1835211)
Affinity DataIC50: 59nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355102(CHEMBL1835325)
Affinity DataIC50: 60nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355099(CHEMBL1835322)
Affinity DataIC50: 86nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355111(CHEMBL1835210)
Affinity DataIC50: 92nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355112(CHEMBL1835211)
Affinity DataIC50: 108nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355097(CHEMBL1835320)
Affinity DataIC50: 136nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355098(CHEMBL1835321)
Affinity DataIC50: 150nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355107(CHEMBL1835403)
Affinity DataIC50: 163nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355093(CHEMBL1835316)
Affinity DataIC50: 219nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355101(CHEMBL1835324)
Affinity DataIC50: 233nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355089(CHEMBL1835212)
Affinity DataIC50: 246nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355098(CHEMBL1835321)
Affinity DataIC50: 289nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355109(CHEMBL1835209)
Affinity DataIC50: 346nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355090(CHEMBL1835313)
Affinity DataIC50: 413nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355110(CHEMBL1835208)
Affinity DataIC50: 437nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355095(CHEMBL1835318)
Affinity DataIC50: 441nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355091(CHEMBL1835314)
Affinity DataIC50: 453nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355106(CHEMBL1835402)
Affinity DataIC50: 459nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355108(CHEMBL1835404)
Affinity DataIC50: 573nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355111(CHEMBL1835210)
Affinity DataIC50: 635nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355092(CHEMBL1835315)
Affinity DataIC50: 772nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355098(CHEMBL1835321)
Affinity DataIC50: 781nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355107(CHEMBL1835403)
Affinity DataIC50: 907nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355112(CHEMBL1835211)
Affinity DataIC50: 965nMAssay Description:Inhibition of C-terminal FLAG-tagged human caspase-3 expressed in HEK293 T17 cells using Ac-DEVD-AMC coumarin-120 as substrate pre-incubated for 2 hr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355108(CHEMBL1835404)
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355099(CHEMBL1835322)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355109(CHEMBL1835209)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355102(CHEMBL1835325)
Affinity DataIC50: 1.41E+3nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355096(CHEMBL1835319)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355110(CHEMBL1835208)
Affinity DataIC50: 1.69E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355112(CHEMBL1835211)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355105(CHEMBL1835401)
Affinity DataIC50: 1.98E+3nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355104(CHEMBL1835400)
Affinity DataIC50: 2.19E+3nMAssay Description:Inhibition of caspase-2 (amino acids 170 to 452) using Ac-VDVAD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355101(CHEMBL1835324)
Affinity DataIC50: 2.26E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355094(CHEMBL1835317)
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355096(CHEMBL1835319)
Affinity DataIC50: 2.77E+3nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355094(CHEMBL1835317)
Affinity DataIC50: 2.93E+3nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-3(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355103(CHEMBL1835399)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of C-terminal histidine-tagged caspase-3 using Ac-DEVD-AMC coumarin-120 as substrate after 20 mins by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCaspase-2(Human)
Chdi Management

Curated by ChEMBL
LigandPNGBDBM50355108(CHEMBL1835404)
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of human Myc-DDK tagged caspase-2 expressed in HEK293 T17 cells using Ac-VDVAD-AMC coumarin-120 as substrate pre-incubated for 2 hrs measu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
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