Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50034030
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355759(CHEMBL1911299)
Affinity DataEC50:  2.10E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355760(CHEMBL1911307)
Affinity DataEC50:  4.10E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50370232(BA-41166E | L-5103 | Rifadin | Rifampicin | RIFAMP...)
Affinity DataEC50:  5.60E+3nMAssay Description:Activation of human PXR in DPX2 cells after 24 hrs by microplate reader relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355756(CHEMBL1909658)
Affinity DataIC50: 13nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355755(CHEMBL1911296)
Affinity DataIC50: 15nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355751(CHEMBL1911286)
Affinity DataIC50: 21nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355758(CHEMBL1911306)
Affinity DataIC50: 139nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355757(CHEMBL1911298)
Affinity DataIC50: 142nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355753(CHEMBL1911289)
Affinity DataIC50: 503nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355752(CHEMBL1911287)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed
TargetDNA-directed RNA polymerase subunit beta(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50355754(CHEMBL1911295)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of wild type Mycobacterium tuberculosis RNA polymerase after 10 mins using ribo green staining by rolling circle transcription assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/20/2012
Entry Details Article
PubMed