Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50033948
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354404(CHEMBL1836407)
Affinity DataKi:  1nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354402(CHEMBL1836405)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354398(CHEMBL1836401)
Affinity DataKi:  1.20nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354401(CHEMBL1836404)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354399(CHEMBL1836402)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354403(CHEMBL1836406)
Affinity DataKi:  1.70nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354400(CHEMBL1836403)
Affinity DataKi:  5.80nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354398(CHEMBL1836401)
Affinity DataKi:  6.5nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354401(CHEMBL1836404)
Affinity DataKi:  6.90nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354403(CHEMBL1836406)
Affinity DataKi:  9.20nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354396(CHEMBL1836399)
Affinity DataKi:  9.40nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354405(CHEMBL1836408)
Affinity DataKi:  10nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354407(CHEMBL1836410)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  12nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM13063(CHEMBL865 | cid_119607 | Bextra | VLX | 4-(5-methy...)
Affinity DataKi:  13nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataKi:  16nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataKi:  21nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  25nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM13063(CHEMBL865 | cid_119607 | Bextra | VLX | 4-(5-methy...)
Affinity DataKi:  27nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10857(aromatic sulfonamide compound 5 | CHEMBL21 | 4-ami...)
Affinity DataKi:  37nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10883(Dichlorophenamide, DCP | CHEMBL17 | Sulfonamide, 4...)
Affinity DataKi:  38nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM13063(CHEMBL865 | cid_119607 | Bextra | VLX | 4-(5-methy...)
Affinity DataKi:  43nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10883(Dichlorophenamide, DCP | CHEMBL17 | Sulfonamide, 4...)
Affinity DataKi:  50nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10883(Dichlorophenamide, DCP | CHEMBL17 | Sulfonamide, 4...)
Affinity DataKi:  50nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354400(CHEMBL1836403)
Affinity DataKi:  57nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354404(CHEMBL1836407)
Affinity DataKi:  57nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354399(CHEMBL1836402)
Affinity DataKi:  59nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354401(CHEMBL1836404)
Affinity DataKi:  59nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354400(CHEMBL1836403)
Affinity DataKi:  62nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354397(CHEMBL1836400)
Affinity DataKi:  68nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354396(CHEMBL1836399)
Affinity DataKi:  69nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354400(CHEMBL1836403)
Affinity DataKi:  76nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354403(CHEMBL1836406)
Affinity DataKi:  76nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354404(CHEMBL1836407)
Affinity DataKi:  78nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354398(CHEMBL1836401)
Affinity DataKi:  78nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354406(CHEMBL1836409)
Affinity DataKi:  86nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354399(CHEMBL1836402)
Affinity DataKi:  87nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354401(CHEMBL1836404)
Affinity DataKi:  87nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354402(CHEMBL1836405)
Affinity DataKi:  102nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354397(CHEMBL1836400)
Affinity DataKi:  104nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10857(aromatic sulfonamide compound 5 | CHEMBL21 | 4-ami...)
Affinity DataKi:  240nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10880(Acetazolamide, AAZ | AZA2 | CHEMBL20 | Acetazolami...)
Affinity DataKi:  250nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarbonic anhydrase 9(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10857(aromatic sulfonamide compound 5 | CHEMBL21 | 4-ami...)
Affinity DataKi:  294nMAssay Description:Inhibition of human carbonic anhydrase 9-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 12(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354402(CHEMBL1836405)
Affinity DataKi:  410nMAssay Description:Inhibition of human carbonic anhydrase 12-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 1(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM10883(Dichlorophenamide, DCP | CHEMBL17 | Sulfonamide, 4...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human carbonic anhydrase 1-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354402(CHEMBL1836405)
Affinity DataKi:  1.71E+3nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354404(CHEMBL1836407)
Affinity DataKi:  2.14E+3nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCarbonic anhydrase 2(Human)
University of Alberta

Curated by ChEMBL
LigandPNGBDBM50354407(CHEMBL1836410)
Affinity DataKi:  4.13E+3nMAssay Description:Inhibition of human carbonic anhydrase 2-catalyzed CO2 hydration activity by stopped flow assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
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