Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50033747
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350660BDBM50350660(CHEMBL1813552)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350661BDBM50350661(CHEMBL1813553)
Affinity DataIC50: 2.70E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350666BDBM50350666(CHEMBL1813558)
Affinity DataIC50: 3.40E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350659BDBM50350659(CHEMBL1813551)
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350669BDBM50350669(CHEMBL1813546)
Affinity DataIC50: 4.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350649BDBM50350649(CHEMBL1813536)
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350670BDBM50350670(CHEMBL1813559)
Affinity DataIC50: 5.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350653BDBM50350653(CHEMBL1813540)
Affinity DataIC50: 5.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350648BDBM50350648(CHEMBL1813535)
Affinity DataIC50: 6.10E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350654BDBM50350654(CHEMBL1813541)
Affinity DataIC50: 6.20E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350657BDBM50350657(CHEMBL1813547)
Affinity DataIC50: 6.50E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350650BDBM50350650(CHEMBL1813537)
Affinity DataIC50: 7.30E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350668BDBM50350668(CHEMBL1813545)
Affinity DataIC50: 8.90E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350652BDBM50350652(CHEMBL1813539)
Affinity DataIC50: 9.80E+3nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350665BDBM50350665(CHEMBL1813557)
Affinity DataIC50: 1.10E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350662BDBM50350662(CHEMBL1813554)
Affinity DataIC50: 1.47E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350647BDBM50350647(CHEMBL1813534)
Affinity DataIC50: 1.80E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350664BDBM50350664(CHEMBL1813556)
Affinity DataIC50: 3.30E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350658BDBM50350658(CHEMBL1813550)
Affinity DataIC50: 3.50E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350656BDBM50350656(CHEMBL1813544)
Affinity DataIC50: 5.20E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350651BDBM50350651(CHEMBL1813538)
Affinity DataIC50: 6.30E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350663BDBM50350663(CHEMBL1813555)
Affinity DataIC50: 6.80E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350655BDBM50350655(CHEMBL1813542)
Affinity DataIC50: 7.50E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350646BDBM50350646(CHEMBL1813533)
Affinity DataIC50: 7.60E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350667BDBM50350667(CHEMBL1813560)
Affinity DataIC50: 8.60E+4nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetTranscriptional activator protein LuxR(Vibrio fischeri)
Insa Lyon

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50350645BDBM50350645(CHEMBL1813532)
Affinity DataIC50: 1.53E+5nMAssay Description:Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescenceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed