Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50035896
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  0.0900nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013847(CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzy...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013849(CHEMBL314209 | 14-[4-azido(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013857(CHEMBL311995 | 14-[4-diazo(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.600nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013857(CHEMBL311995 | 14-[4-diazo(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013847(CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzy...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013849(CHEMBL314209 | 14-[4-azido(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013849(CHEMBL314209 | 14-[4-azido(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013849(CHEMBL314209 | 14-[4-azido(methyl)anilino]-4-cyclo...)
Affinity DataKi:  0.700nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013857(CHEMBL311995 | 14-[4-diazo(methyl)anilino]-4-cyclo...)
Affinity DataKi:  1nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013857(CHEMBL311995 | 14-[4-diazo(methyl)anilino]-4-cyclo...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013855(CHEMBL312046 | 1-(4-Azido-phenyl)-8-[1-(4-chloro-p...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013848(CHEMBL312281 | 8-[1-(4-Chloro-phenyl)-ethyl]-1-phe...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013855(CHEMBL312046 | 1-(4-Azido-phenyl)-8-[1-(4-chloro-p...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  6.70nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013853(CHEMBL81328 | 1-[2-(4-Azido-phenyl)-ethyl]-4-(phen...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013853(CHEMBL81328 | 1-[2-(4-Azido-phenyl)-ethyl]-4-(phen...)
Affinity DataKi:  8nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM60212(SMR000058767 | NALTREXONE HYDROCHLORIDE | MLS00006...)
Affinity DataKi:  8.70nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  9nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013848(CHEMBL312281 | 8-[1-(4-Chloro-phenyl)-ethyl]-1-phe...)
Affinity DataKi:  10nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013852(CHEMBL81465 | 1-(2-Diethylamino-ethyl)-2-(4-ethoxy...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013850(CHEMBL84237 | 4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-o...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013852(CHEMBL81465 | 1-(2-Diethylamino-ethyl)-2-(4-ethoxy...)
Affinity DataKi:  18nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013856(CHEMBL309542 | 1-[2-(4-Azido-3-iodo-phenyl)-ethyl]...)
Affinity DataKi:  27nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013856(CHEMBL309542 | 1-[2-(4-Azido-3-iodo-phenyl)-ethyl]...)
Affinity DataKi:  45nMAssay Description:Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
LigandPNGBDBM50013850(CHEMBL84237 | 4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-o...)
Affinity DataKi:  62nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013848(CHEMBL312281 | 8-[1-(4-Chloro-phenyl)-ethyl]-1-phe...)
Affinity DataKi:  75nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50012477(1-Phenethyl-4-(phenyl-propionyl-amino)-piperidine-...)
Affinity DataKi:  92nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013855(CHEMBL312046 | 1-(4-Azido-phenyl)-8-[1-(4-chloro-p...)
Affinity DataKi:  100nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  242nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013854(CHEMBL310829 | {2-[5-Azido-2-(4-ethoxy-benzyl)-ben...)
Affinity DataKi:  400nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013856(CHEMBL309542 | 1-[2-(4-Azido-3-iodo-phenyl)-ethyl]...)
Affinity DataKi: >1.00E+3nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013847(CHEMBL312040 | Etonitazene | {2-[2-(4-Ethoxy-benzy...)
Affinity DataKi: >1.00E+3nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013853(CHEMBL81328 | 1-[2-(4-Azido-phenyl)-ethyl]-4-(phen...)
Affinity DataKi: >1.00E+3nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013850(CHEMBL84237 | 4-{8-[1-(4-Chloro-phenyl)-ethyl]-4-o...)
Affinity DataKi: >1.00E+3nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013853(CHEMBL81328 | 1-[2-(4-Azido-phenyl)-ethyl]-4-(phen...)
Affinity DataKi: >1.00E+3nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013852(CHEMBL81465 | 1-(2-Diethylamino-ethyl)-2-(4-ethoxy...)
Affinity DataKi: >1.00E+4nMAssay Description:Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50013856(CHEMBL309542 | 1-[2-(4-Azido-3-iodo-phenyl)-ethyl]...)
Affinity DataKi: >1.00E+4nMAssay Description:Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2012
Entry Details Article
PubMed