Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50034463
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50312315(PEPTAPPEE | CHEMBL1075925)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to Tsg101More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human Tsg101 binding to GST-tagged P6 protein by surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362889(CHEMBL1946129)
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of human Tsg101 binding to GST-tagged P6 protein by surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362892(CHEMBL1946564)
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362891(CHEMBL1946260)
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362890(CHEMBL1946259)
Affinity DataKi:  5.40E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetTumor susceptibility gene 101 protein(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50362889(CHEMBL1946129)
Affinity DataKi:  8.70E+3nMAssay Description:Displacement of FITC-conjugated (S)-4-((S)-1-acetylpyrrolidine-2-carboxamido)-5-((2S,4R)-2-((2S,3R)-1-((S)-1-((S)-2-((S)-2-((S)-1-((S)-1-amino-4-carb...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed