Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50033424
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345056(2-(6-(3-((dimethylamino)methyl)phenyl)-2-(4-fluoro...)
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345045(N-isopropyl-2-(2-(3-methoxyphenyl)-4-oxo-6-(3-(pip...)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345055(2-(6-(5-((dimethylamino)methyl)-2-fluorophenyl)-2-...)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345048(2-(2-(3-chlorophenyl)-4-oxo-6-(3-(piperidin-1-ylme...)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345043(2-(6-(3-((dimethylamino)methyl)phenyl)-2-(3-methox...)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345046(2-(2-(3-chlorophenyl)-6-(3-((dimethylamino)methyl)...)
Affinity DataIC50: 19nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345052(2-(6-(6-((dimethylamino)methyl)pyridin-2-yl)-2-(3-...)
Affinity DataIC50: 37nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345044(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(3-methoxyp...)
Affinity DataIC50: 46nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345050(2-(6-(4-((dimethylamino)methyl)pyridin-2-yl)-2-(3-...)
Affinity DataIC50: 52nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345060(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(3-(pipe...)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345047(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(3-chloroph...)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345051(2-(6-(5-((dimethylamino)methyl)pyridin-3-yl)-2-(3-...)
Affinity DataIC50: 77nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345059(N-(cyclopropylmethyl)-2-(6-(3-(morpholinomethyl)ph...)
Affinity DataIC50: 79nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345040(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 187nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345042(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 238nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345034(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 275nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345032(N-(cyclopropylmethyl)-2-(6-(3-((dimethylamino)meth...)
Affinity DataIC50: 314nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345064(N-(cyclopropylmethyl)-2-(6-(3-((methylamino)methyl...)
Affinity DataIC50: 320nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345035(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(3-(pyrr...)
Affinity DataIC50: 388nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345039(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 397nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345054(2-(6-(5-((dimethylamino)methyl)thiophen-2-yl)-2-(3...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345033(N-(cyclopropylmethyl)-2-(6-(3-((diethylamino)methy...)
Affinity DataIC50: 540nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345049(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-2-(2-methoxyp...)
Affinity DataIC50: 610nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345036(N-(cyclopropylmethyl)-2-(6-(3-((2-methoxyethylamin...)
Affinity DataIC50: 642nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345053(2-(6-(5-((dimethylamino)methyl)furan-2-yl)-2-(3-me...)
Affinity DataIC50: 700nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345038(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345063(2-(6-(3-(aminomethyl)phenyl)-4-oxo-2-phenylquinazo...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345037(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 2.35E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345041(2-(6-(3-(azetidin-1-ylmethyl)phenyl)-4-oxo-2-pheny...)
Affinity DataIC50: 2.55E+3nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345057(N-(cyclopropylmethyl)-2-(6-(2-(morpholinomethyl)ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345058(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(2-(pipe...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345061(N-(cyclopropylmethyl)-2-(6-(4-(morpholinomethyl)ph...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetVasopressin V1b receptor(Human)
Msd

Curated by ChEMBL
LigandPNGBDBM50345062(N-(cyclopropylmethyl)-2-(4-oxo-2-phenyl-6-(4-(pipe...)
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of [3H]AVP from human vasopressin V1b receptor expressed in CHO cells co-expressing VIP-luciferase by scintillation counting-based whole...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed