Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50033418
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50299505(3 9-dihydro-N-desmethyl-N-isopropylerythromycin A ...)
Affinity DataEC50:  260nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Human)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | ERYTHROMYCIN | Erycette | Erymax | Ery...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at motilin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50299502(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  660nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50299517(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  58nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50299518(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  52nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344956((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344955((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  360nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344954((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  210nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344953((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-6-((2S,3R,...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344942(CHEMBL532 | ERYTHROMYCIN | Erycette | Erymax | Ery...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344952((2R,3S,4R,5R,8R,9S,10S,11R,12S)-5-ethyl-11-((2S,3R...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344951(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344950(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344949(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataEC50:  36nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344948((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344947((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344946(2-(((2S,3R,4S,6R)-2-((3R,4S,5S,6R,7R,9R,10S,11S,12...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344945((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  63nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344944((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-6-((2S,3R,...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetMotilin receptor(Rabbit)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344943((3R,4S,5S,6R,7R,9R,10S,11S,12R,13S,14R)-14-ethyl-7...)
Affinity DataEC50:  59nMAssay Description:Agonist activity at motilin receptor in rabbit smooth muscle assessed as maximal possible tissue contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50344950(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Kosan Biosciences

Curated by ChEMBL
LigandPNGBDBM50299517(2-((2R,3S,4R,5R,6S,7R,9R,10R,11S,12S,13R)-2-ethyl-...)
Affinity DataIC50: 4.11E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed