Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50033757
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350763(CHEMBL1818445)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CYP2C9 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350763(CHEMBL1818445)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CYP2C19 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350763(CHEMBL1818445)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CYP3A4 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350763(CHEMBL1818445)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CYP2D6 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350763(CHEMBL1818445)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human CYP1A2 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350766(CHEMBL1818455)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human CYP2D6 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350766(CHEMBL1818455)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human CYP2C9 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350766(CHEMBL1818455)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human CYP1A2 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350766(CHEMBL1818455)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human CYP3A4 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350766(CHEMBL1818455)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human CYP2C19 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350764(CHEMBL1818451)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2D6 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350765(CHEMBL1818452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP3A4 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350764(CHEMBL1818451)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP3A4 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350765(CHEMBL1818452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2D6 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350765(CHEMBL1818452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2C19 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350764(CHEMBL1818451)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2C19 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350765(CHEMBL1818452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2C9 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350764(CHEMBL1818451)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP2C9 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350765(CHEMBL1818452)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP1A2 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350764(CHEMBL1818451)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CYP1A2 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C9(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350767(CHEMBL1818543)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CYP2C9 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350767(CHEMBL1818543)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CYP2C19 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350767(CHEMBL1818543)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CYP2D6 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350767(CHEMBL1818543)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CYP3A4 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 1A2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50350767(CHEMBL1818543)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human CYP1A2 incubated for 10 mins before substrate addition by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed