Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50033450
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345577(Hippolide A | CHEMBL1782082)
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetTyrosine-protein phosphatase non-receptor type 1(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345576(Hippolide B | CHEMBL1784622)
Affinity DataIC50: 3.97E+4nMAssay Description:Inhibition of recombinant PTP1B catalytic domain using pNPP as substrate assessed as pNP releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345578(Hippolide E | CHEMBL1784623)
Affinity DataIC50: 4.04E+4nMAssay Description:Binding affinity at PKCalpha after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50345577(Hippolide A | CHEMBL1782082)
Affinity DataIC50: 6.20E+4nMAssay Description:Binding affinity at PKCgamma after 1 hr by luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed