Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50033393
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50301022((+)-9-fluoropropyl-dihydrotetrabenazine | CHEMBL57...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50301021((+)-dihydrotetrabenzaine | CHEMBL576222 | US110532...)
Affinity DataKi:  1.03nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344439(rac-(2R)-9,10-dimethoxy-3-(2-methylallyl)-2,3,4,6,...)
Affinity DataKi:  5.98nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344443(rac-(2R)-9-(3-fluoropropoxy)-10-methoxy-3-(prop-1-...)
Affinity DataKi:  22.4nMAssay Description:Displacement of [18F](+)-FP-DTBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344440(rac-(2R)-3-(cyclobutylmethyl)-9,10-dimethoxy-2,3,4...)
Affinity DataKi:  26.9nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344442(rac-(2R)-3-(cyclohexylmethyl)-9,10-dimethoxy-2,3,4...)
Affinity DataKi:  137nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344441(rac-(2R)-3-(cyclopentylmethyl)-9,10-dimethoxy-2,3,...)
Affinity DataKi:  227nMAssay Description:Displacement of [125I]-iodovinyl-TBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetSynaptic vesicular amine transporter(Rat)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50344438(rac-(2R)-3-allyl-9,10-dimethoxy-2,3,4,6,7,11b-hexa...)
Affinity DataKi:  253nMAssay Description:Displacement of [18F](+)-FP-DTBZ from VMAT2 in rat striatal homogenate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed