Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50033430
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM13061(CHEMBL1444 | 4-[(4-cyanophenyl)(1H-1,2,4-triazol-1...)
Affinity DataIC50: 18nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345191(7,8-Benzo-4'-hydroxy-4-imidazolylflavan | CHEMBL17...)
Affinity DataIC50: 32nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50: 34nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345189(2,4-trans-7,8-benzo-4-imidazolylflavan | CHEMBL178...)
Affinity DataIC50: 36nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50: 60nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50: 91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50118966(1-(7-Methoxy-2-phenyl-chroman-4-yl)-1H-imidazole |...)
Affinity DataIC50: 91nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50: 534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345190(2,4-cis-7,8-benzo-4'-cyano-4-imidazolylflavan | 2,...)
Affinity DataIC50: 534nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345188(2-(4-hydroxyphenyl)-2,3-dihydrobenzo[h]chromen-4-o...)
Affinity DataIC50: 630nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345187(4-(4-oxo-3,4-dihydro-2H-benzo[h]chromen-2-yl)benzo...)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM50345186(2-phenyl-2,3-dihydrobenzo[h]chromen-4-one | 2-phen...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetAromatase(Human)
Upres Ea 4021 Biomol�Cules Et Th�Rapies Anti-Tumorales

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | C...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of aromatase in human placental microsomes assessed as inhibition of aromatization of [1,2,6,7-3H] androstenedione by flow scintillation a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed