Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50033261
TargetMitogen-activated protein kinase 9(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataKd:  640nMAssay Description:Binding affinity to JNK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to JNK1 in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to JNK1 in presence of peptide JIP1More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342302(2-(2-(2-chlorophenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342305(2-(2-(3-iodophenyl)acetamido)thiophene-3-carboxami...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342304(2-(2-(3-bromophenyl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342303(2-(2-(benzo[d][1,3]dioxol-5-yl)acetamido)thiophene...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342306(2-(2-(4-ethoxyphenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342307(2-(2-(9-chloro-3,4-dihydro-2H-benzo[b][1,4]dioxepi...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342308(2-(2-(2-methoxy-5-methylphenyl)acetamido)thiophene...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342309(2-(2-(2,3-dihydro-1H-inden-5-yl)acetamido)thiophen...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342310(2-(2-(6-(thiophen-2-yl)imidazo[2,1-b]thiazol-3-yl)...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342311(2-(2-(5-methylimidazo[2,1-b]thiazol-2-yl)acetamido...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342312(2-(2-(3-chlorophenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342313(2-(2-(3-methoxyphenyl)acetamido)thiophene-3-carbox...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342314(2-(2-(3,5-dimethylphenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342315(2-(2-(2,3-dihydrobenzo[b][1,4]dioxin-6-yl)acetamid...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342316(2-(2-(2-bromophenyl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342317(2-(2-(4-nitrophenyl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342318(2-(2-(3,5-dimethoxyphenyl)acetamido)thiophene-3-ca...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342319(2-(2-(thiophen-2-yl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342320(2-(2-(2-iodophenyl)acetamido)thiophene-3-carboxami...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342321(2-(2-(4-cyanophenyl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342322(2-(2-phenylacetamido)thiophene-3-carboxamide | CHE...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342323(2-(2-(5,6,7,8-tetrahydronaphthalen-2-yl)acetamido)...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342324(2-(2-p-tolylacetamido)thiophene-3-carboxamide | CH...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataIC50: 4.62E+3nMAssay Description:Displacement of biotin-labeled JIP1 peptide from JNK1 by DELFIA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342325(2-(2-(6-fluoro-4H-benzo[d][1,3]dioxin-8-yl)acetami...)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342326(2-(2-(4-fluorophenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342327(2-(2-(naphthalen-1-yl)acetamido)thiophene-3-carbox...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342328(2-(2-m-tolylacetamido)thiophene-3-carboxamide | CH...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342329(2-(2-(4-methoxyphenyl)acetamido)thiophene-3-carbox...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342330(2-(2-(4-(trifluoromethoxy)phenyl)acetamido)thiophe...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342331(2-(2-(2,5-difluorophenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342332(2-benzamidothiophene-3-carboxamide | CHEMBL1767238)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342333(2-(2-o-tolylacetamido)thiophene-3-carboxamide | CH...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342334(2-(2-(4-(trifluoromethyl)phenyl)acetamido)thiophen...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342335(2-(2-(2,6-difluorophenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetTranscription factor Jun(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342301(2-(2-(benzo[b]thiophen-3-yl)acetamido)thiophene-3-...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of TNF-alpha-induced c-Jun phosphorylation in human HeLa cells by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342336(2-(2-(3-(trifluoromethyl)phenyl)acetamido)thiophen...)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342337(2-(2-(4-(furan-2-ylmethyl)piperazin-1-yl)acetamido...)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342338(2-(2-(pyridin-3-yl)acetamido)thiophene-3-carboxami...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342339(2-(2-(3,5-difluorophenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342340(2-(2-(2-fluorophenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342341(2-(2-(3-fluorophenyl)acetamido)thiophene-3-carboxa...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342342(2-(2-(1H-indol-3-yl)acetamido)thiophene-3-carboxam...)
Affinity DataIC50: 9.40E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342343(2-(2-(2,4-difluorophenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342344(2-(2-(3,4-difluorophenyl)acetamido)thiophene-3-car...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50342345(2-(2-(2-methoxyphenyl)acetamido)thiophene-3-carbox...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of JNK1 by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
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