Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50033242
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(Voglibose | CHEMBL476960)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(Salaprinol | CHEMBL1209027)
Affinity DataIC50: 290nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50: 750nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(Voglibose | CHEMBL476960)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5S,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5S,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50263044(Voglibose | CHEMBL476960)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(Salaprinol | CHEMBL1209027)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50338672(Salaprinol | CHEMBL1209027)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50330955((1S,2S)-3-[(2R,3S,4S)-3,4-dihydroxy-2-(hydroxymeth...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50316179((1S,2R,3R,4S)-1-{(1S)-2-[(2R,3S,4S)-3,4-dihydroxy-...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341973(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341975(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341972(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341974(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341974(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341974(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50327501(ponkoranol | CHEMBL1258528)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50327501(ponkoranol | CHEMBL1258528)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50333465((2R,3R,4R,5S,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50: 1.55E+5nMAssay Description:Inhibition of rat small intestinal isomaltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341975(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341972(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341972(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5S,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341973(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetSucrase-isomaltase, intestinal(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341975(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6R)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal sucrase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLysosomal alpha-glucosidase(Rat)
Kinki University

Curated by ChEMBL
LigandPNGBDBM50341973(1,4-dideoxy-1,4-{(S)-[(2S,3R,4S,5R,6S)-2,4,5,6,7-p...)
Affinity DataIC50: 2.36E+5nMAssay Description:Inhibition of rat small intestinal maltase after 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed