Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 50033141
LigandPNGBDBM16673(Xarelto | BAY439006 | CHEMBL1336 | BAY 43-9006 | 4...)
Affinity DataIC50: 40nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340266(7-(2-(3-(4-chloro-2-methoxy-5-(trifluoromethyl)phe...)
Affinity DataIC50: 80nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340264(7-(2-(3-(5-chloro-2-methoxy-4-methylphenyl)ureido)...)
Affinity DataIC50: 110nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340262(7-(2-(3-(2-methoxy-5-(trifluoromethyl)phenyl)ureid...)
Affinity DataIC50: 120nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340273(N-(6-(2-(3-(4-chloro-3-(trifluoromethyl)phenyl)ure...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340259(7-(2-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340270(N-(6-(2-(3-(2-methoxy-5-(trifluoromethyl)phenyl)ur...)
Affinity DataIC50: 170nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340285(N-(6-(2-(3-(2-(2-aminoethoxy)-4-chloro-5-(trifluor...)
Affinity DataIC50: 180nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340265(7-(2-(3-(4-chloro-2-methoxy-5-methylphenyl)ureido)...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340277(N-(6-(2-(3-(5-chloro-2-methoxy-4-methylphenyl)urei...)
Affinity DataIC50: 190nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340258(N-methyl-7-(2-(3-(4-methyl-3-(trifluoromethyl)phen...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340288(N-methyl-7-(2-(3-(3-(trifluoromethylsulfonyl)pheny...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340281(N-(6-(2-(3-(2-(2-(methylamino)ethoxy)-5-(trifluoro...)
Affinity DataIC50: 210nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340290(N-(6-(2-(3-(2-(pyrrolidin-2-ylmethoxy)-5-(trifluor...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340282(N-(6-(2-(3-(4-chloro-2-(2-(methylamino)ethoxy)-5-(...)
Affinity DataIC50: 230nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340260(7-(2-(3-(4-fluoro-3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 240nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340261(7-(2-(3-(2-fluoro-5-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340284(N-(6-(2-(3-(2-(2-aminoethoxy)-5-(trifluoromethyl)p...)
Affinity DataIC50: 250nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340287(N-methyl-7-(2-(3-(3-(trifluoromethoxy)phenyl)ureid...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340271(6-(2-(3-(4-chloro-3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 280nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340278(N-(6-(2-(3-(4-chloro-2-methoxy-5-methylphenyl)urei...)
Affinity DataIC50: 320nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340268(6-(2-(3-(2-methoxy-5-(trifluoromethyl)phenyl)ureid...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340267(7-(2-(3-(4-chloro-2-(2-(dimethylamino)ethoxy)-5-(t...)
Affinity DataIC50: 340nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340286(N-methyl-7-(2-(3-(3-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 360nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340289(N-methyl-7-(2-(3-(4-(trifluoromethyl)phenyl)ureido...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340263(7-(2-(3-(2-(2-(dimethylamino)ethoxy)-5-(trifluorom...)
Affinity DataIC50: 450nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340275(N-(6-(2-(3-(3,4-dichlorophenyl)ureido)ethyl)-1H-be...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340274(N-(6-(2-(3-(3-(trifluoromethyl)phenyl)ureido)ethyl...)
Affinity DataIC50: 480nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340280(N-(6-(2-(3-(4-chloro-5-methyl-2-(2-(methylamino)et...)
Affinity DataIC50: 490nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340276(N-(6-(2-(3-(3-chloro-4-methylphenyl)ureido)ethyl)-...)
Affinity DataIC50: 530nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340283(N-(6-(2-(3-(2-(2-aminoethoxy)-4-chloro-5-methylphe...)
Affinity DataIC50: 550nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340279(N-(6-(2-(3-(5-methyl-2-(2-(methylamino)ethoxy)phen...)
Affinity DataIC50: 580nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340272(methyl 6-(2-(3-(4-chloro-3-(trifluoromethyl)phenyl...)
Affinity DataIC50: 660nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
LigandPNGBDBM50340269(methyl 6-(2-(3-(2-methoxy-5-(trifluoromethyl)pheny...)
Affinity DataIC50: 810nMAssay Description:Inhibition of human cRAF using [gamma-33P-ATP] as a substrate by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed