Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50033233
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataKd:  1.00E+4nMAssay Description:Displacement of FAM-AHA-ARTKQTARK(Me)STGGKA-CO2H from human L3MBTL1 assessed as apparent dissociation constant after 20 mins by FP-displacement AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341829(3-Bromo-N-(5-pyrrolidin-1-yl)pentylbenzenesulfonam...)
Affinity DataKd:  2.50E+4nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341830(5-Bromo-N-(5-(pyrrolidin-1-yl)pentylnicotinamide |...)
Affinity DataKd:  2.60E+4nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341831((S)-2-amino-3-(1H-imidazol-4-yl)-N-((S)-1-oxo-3-ph...)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341832((S)-3-Bromo-N-(5-(3-fluoro)pyrrolidin-1-yl)pentylb...)
Affinity DataKd:  5.10E+4nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341833((S)-2-amino-N-((S)-1-(5-(ethyl(methyl)amino)pentyl...)
Affinity DataKd:  7.80E+4nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341834((S)-2-amino-3-(1H-imidazol-4-yl)-N-((S)-1-(5-(meth...)
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341835((S)-2-amino-N-((S)-1-(5-(dimethylamino)pentylamino...)
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341836(5-Bromo-N-(5-(2-methyl)pyrrolidin-1-yl)pentylbenze...)
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to human L3MBTL1 assessed as dissociation constant by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50: 6.00E+3nMAssay Description:Binding affinity to human L3MBTL1 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLethal(3)malignant brain tumor-like protein 3(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341830(5-Bromo-N-(5-(pyrrolidin-1-yl)pentylnicotinamide |...)
Affinity DataIC50: 2.80E+4nMAssay Description:Binding affinity to L3MBTL3 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLethal(3)malignant brain tumor-like protein 3(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50: 3.50E+4nMAssay Description:Binding affinity to L3MBTL3 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetIsoform 4 of Lethal(3)malignant brain tumor-like protein 1 (4)(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341830(5-Bromo-N-(5-(pyrrolidin-1-yl)pentylnicotinamide |...)
Affinity DataIC50: 4.60E+4nMAssay Description:Binding affinity to human L3MBTL1 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetPHD finger protein 13(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341830(5-Bromo-N-(5-(pyrrolidin-1-yl)pentylnicotinamide |...)
Affinity DataIC50: 4.80E+4nMAssay Description:Binding affinity to PHF13 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetLethal(3)malignant brain tumor-like protein 4(Human)
University of North Carolina at Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50: 6.90E+4nMAssay Description:Binding affinity to L3MBTL4 by chemiluminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed