Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50033213
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341487(Succinyl-alaninyl-alaninyl-prolinyl-phenylalaninyl...)
Affinity DataIC50: 0.700nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated with alpha-chymotrypsin up to 8 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 1nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 1.5nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341488(Phenylalaninyl-prolinyl-alaninyl-L-boroproline | C...)
Affinity DataIC50: 7nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341488(Phenylalaninyl-prolinyl-alaninyl-L-boroproline | C...)
Affinity DataIC50: 8.30nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341489(Cyclohexyl(glycinyl)-prolinyl-valinyl-L-boroprolin...)
Affinity DataIC50: 19nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50341489(Cyclohexyl(glycinyl)-prolinyl-valinyl-L-boroprolin...)
Affinity DataIC50: 20nMpH: 2.0Assay Description:Inhibition of DDP4 at pH 2 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050513(Ketopyrrolidine derivative | (R)-1-((S)-2-amino-3-...)
Affinity DataIC50: 470nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Tufts University Sackler School of Graduate Biomedical Sciences

Curated by ChEMBL
LigandPNGBDBM50050525((R)-1-((S)-2-aminopropanoyl)pyrrolidin-2-ylboronic...)
Affinity DataIC50: 1.60E+3nMpH: 7.4Assay Description:Inhibition of DDP4 at pH 7.4 preincubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed