Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50033178
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340946((1R,3S,14S)-6,10,14-trimethyl-3-(prop-1-en-2-yl)-1...)
Affinity DataEC50:  1.08E+5nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340947((6R,8S,18R)-3,8,12,16-Tetramethyl-7,18-dioxa-tricy...)
Affinity DataEC50:  1.83E+5nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340948((1E,3E,7R*,8R*,11E)-1-(2-methoxypropan-2-yl)-4,8,1...)
Affinity DataEC50:  1.49E+5nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340949((1R,2S)-1-((1R,4aS,11aR)-1-acetoxy-7-methyl-11-met...)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340950((1R,2S)-1-((1R,4aS,9R,11aR)-1-acetoxy-9-hydroxy-7-...)
Affinity DataEC50:  6.20E+3nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
TargetEndothelial PAS domain-containing protein 1(Human)
Nci-Frederick

Curated by ChEMBL
LigandPNGBDBM50340951((1R,2S)-1-((1R,4aS,8S,11aR)-1-acetoxy-8-hydroperox...)
Affinity DataEC50:  1.18E+4nMAssay Description:Inhibition of HIF-2alpha activity in human 786-O cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed