Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50033167
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340753(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340743(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340744(N-benzyl-2-(4-(2-(4-chlorophenethylamino)pyrimidin...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340745(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340746(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340750(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 77nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340747(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 88nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340751(N-((3-bromopyridin-4-yl)methyl)-2-(4-(2-(4-chlorop...)
Affinity DataIC50: 108nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340748(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 244nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340749(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 295nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340741(4-(2-(2-(4-chlorophenethylamino)pyrimidin-4-ylamin...)
Affinity DataIC50: 301nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340752(N-benzyl-2-(4-(2-(4-chlorophenethylamino)pyrimidin...)
Affinity DataIC50: 330nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340738(1-(2-(4-chlorophenethylamino)-4-(pyrrolidin-1-yl)q...)
Affinity DataIC50: 530nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340740(4-(2-(2-(4-chlorophenethylamino)quinazolin-4-ylami...)
Affinity DataIC50: 640nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340742(2-(4-(2-(4-chlorophenethylamino)pyrimidin-4-yl)pip...)
Affinity DataIC50: 758nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed
TargetMas-related G-protein coupled receptor member X1(Human)
Astrazeneca R&D Montreal

Curated by ChEMBL
LigandPNGBDBM50340739(N-(4-chlorophenethyl)-4-(pyrrolidin-1-yl)quinazoli...)
Affinity DataIC50: 8.06E+3nMAssay Description:Antagonist activity at SNSR4 in human HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed