Compile Data Set for Download or QSAR
Report error Found 81 Enz. Inhib. hit(s) with all data for entry = 50033012
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338099(3-(6-methyl-1H-indol-2-yl)-N-(1-methylpiperidin-4-...)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338098(3-(6-methyl-1H-indol-2-yl)-N-(piperidin-4-yl)-1H-i...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338077(2-(1H-indazol-3-yl)-N-isobutyl-N-methyl-1H-indole-...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338079(2-(1H-indazol-3-yl)-N-((1-methyl-1H-imidazol-5-yl)...)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338100(N-(1-benzylpiperidin-4-yl)-3-(6-methyl-1H-indol-2-...)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338056(1-methyl-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338058(N1,N1-dimethyl-N2-(3-(6-methyl-1H-indol-2-yl)-1H-i...)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338112(N-(1-benzylpyrrolidin-3-yl)-3-(6-methyl-1H-indol-2...)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338049(N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-5-yl)meth...)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338057(1,5-dimethyl-N-(3-(6-methyl-1H-indol-2-yl)-1H-inda...)
Affinity DataIC50: 43nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338052(3-fluoro-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-...)
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338054(3-methoxy-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol...)
Affinity DataIC50: 46nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338051(2-fluoro-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-...)
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338117(2-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338074(N-benzyl-2-(1H-indazol-3-yl)-N-methyl-1H-indole-6-...)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50331277(3-(6-methoxy-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyri...)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338105(2-(dimethylamino)-N-(3-(6-methyl-1H-indol-2-yl)-1H...)
Affinity DataIC50: 65nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338115(N-(1-ethylpiperidin-3-yl)-3-(6-methyl-1H-indol-2-y...)
Affinity DataIC50: 66nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338103(N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-5-yl)acet...)
Affinity DataIC50: 67nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338050(N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-5-yl)benz...)
Affinity DataIC50: 69nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338076(2-(1H-indazol-3-yl)-N-(2-methoxyethyl)-N-methyl-1H...)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338075(N,N-diethyl-2-(1H-indazol-3-yl)-1H-indole-6-carbox...)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338080(3-(6-(2-methoxyethyl)-1H-indol-2-yl)-1H-pyrazolo[4...)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338088(1-(3,5-dimethylisoxazol-4-yl)-3-(3-(6-methyl-1H-in...)
Affinity DataIC50: 72nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338114(3-(6-methyl-1H-indol-2-yl)-N-(piperidin-3-yl)-1H-i...)
Affinity DataIC50: 77nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338116(3-(6-methyl-1H-indol-2-yl)-N-(pyrrolidin-3-yl)-1H-...)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338085(1-ethyl-3-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-5...)
Affinity DataIC50: 83nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338110(1,3,5-trimethyl-N-(3-(6-methyl-1H-indol-2-yl)-1H-i...)
Affinity DataIC50: 85nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338045(N-(3-(6-methoxy-1H-indol-2-yl)-1H-indazol-5-yl)ace...)
Affinity DataIC50: 87nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338046(2-methoxy-N-(3-(6-methoxy-1H-indol-2-yl)-1H-indazo...)
Affinity DataIC50: 98nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338073(N-benzyl-2-(1H-indazol-3-yl)-1H-indole-6-carboxami...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338101(1-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338102(2-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 100nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338065(3-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338078(N-(furan-2-ylmethyl)-2-(1H-indazol-3-yl)-N-methyl-...)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338104(2-methoxy-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol...)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338070(4-(2-(1H-indazol-3-yl)-1H-indol-6-yl)morpholine | ...)
Affinity DataIC50: 120nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338118(3,5-dimethyl-N-(3-(6-methyl-1H-indol-2-yl)-1H-inda...)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338041(N-(3-(1H-indol-2-yl)-1H-indazol-5-yl)acetamide | C...)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338063(3-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 140nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338042(N-(3-(1H-indol-2-yl)-1H-indazol-5-yl)-2-methoxyace...)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338111(2,4-dimethyl-N-(3-(6-methyl-1H-indol-2-yl)-1H-inda...)
Affinity DataIC50: 190nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338072(N-(cyclohexylmethyl)-2-(1H-indazol-3-yl)-1H-indole...)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338084(3-(6-benzyl-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyrid...)
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338059(N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-6-yl)acet...)
Affinity DataIC50: 220nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338053(4-fluoro-N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-...)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338068(2-(1H-indazol-3-yl)-N-(2-methoxyethyl)-1H-indol-6-...)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338107(N-(3-(6-methyl-1H-indol-2-yl)-1H-indazol-5-yl)tetr...)
Affinity DataIC50: 260nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338064(3-(6-(3-methoxyprop-1-ynyl)-1H-indol-2-yl)-1H-pyra...)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Nycomed

Curated by ChEMBL
LigandPNGBDBM50338066(3-(2-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1H-indol-6-y...)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant GST-tagged full-length ITK expressed in baculovirus expression system after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
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