Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50033005
LigandPNGBDBM50337887((S)-1-methylcyclopropyl 4-(1-fluoro-2-(2-(2,3,6-tr...)
Affinity DataEC50:  80nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337888(tert-butyl 4-(1-(2-(2,3,6-trifluorophenyl)acetamid...)
Affinity DataEC50:  13nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337889(tert-butyl 4-(1-(2-(4-(methylsulfonyl)phenyl)aceta...)
Affinity DataEC50:  884nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337890(tert-butyl 4-(1-(2-(4-(1H-tetrazol-1-yl)phenyl)ace...)
Affinity DataEC50:  267nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337891(tert-butyl 4-(1-(2-(2,3-difluorophenyl)acetamido)p...)
Affinity DataEC50:  75nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337892(tert-butyl 4-(1-(2-(2,5-difluorophenyl)acetamido)p...)
Affinity DataEC50:  78nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337893(tert-butyl 4-(1-(2-(2,6-difluorophenyl)acetamido)p...)
Affinity DataEC50:  120nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337894(tert-butyl 4-(1-(2-(2-fluorophenyl)acetamido)propa...)
Affinity DataEC50:  808nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337895(tert-butyl 4-(1-(2-(3-fluorophenyl)acetamido)propa...)
Affinity DataEC50:  340nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337896(tert-butyl 4-(1-(2-phenylacetamido)propan-2-yl)pip...)
Affinity DataEC50:  5.98E+3nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337897(isopropyl 4-(1-(2-(2,3,6-trifluorophenyl)acetamido...)
Affinity DataEC50:  32nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337899(isopropyl 4-(2-(2-(2,3,6-trifluorophenyl)acetamido...)
Affinity DataEC50:  409nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337900((R)-1-methylcyclopropyl 4-(1-fluoro-2-(2-(2,3,6-tr...)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50337901(1-methylcyclopropyl 4-(2-(2-(2,3,6-trifluorophenyl...)
Affinity DataEC50:  868nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50418004(CHEMBL2092727)
Affinity DataEC50:  44nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
LigandPNGBDBM50418005(CHEMBL2092875)
Affinity DataEC50:  236nMAssay Description:Agonist activity against human GPR119 receptor expressed in HEK293 cells assessed as beta-lactamase production by cAMP response element assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed