Compile Data Set for Download or QSAR
Report error Found 71 Enz. Inhib. hit(s) with all data for entry = 50032975
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337251((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)
Affinity DataIC50: 0.200nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337251((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)
Affinity DataIC50: 1.10nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337250((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 1.20nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337251((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337236((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 2.30nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337238((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337242((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337212(5-chloro-6-((3S)-4-(1-(1-(4-chlorophenyl)ethyl)pip...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337212(5-chloro-6-((3S)-4-(1-(1-(4-chlorophenyl)ethyl)pip...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337237((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 6.70nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337233((S)-N-(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-...)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 9.90nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337219((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337210((S)-5-chloro-6-(4-(1-(2,4-dichlorobenzyl)piperidin...)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337262((S)-5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)pipe...)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337234((S)-N-(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337239((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337218((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human CXCR3 by chemotaxis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337252((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337224(5-chloro-6-(4-(1-(4-chlorobenzyl)-4-methylpiperidi...)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337213(5-chloro-6-((3S)-4-(1-(5-chloro-2,3-dihydro-1H-ind...)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337213(5-chloro-6-((3S)-4-(1-(5-chloro-2,3-dihydro-1H-ind...)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50301330(5-chloro-6-(4-((2S)-1-(4-chlorobenzyl)-2-methylpip...)
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337254((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337253(5-chloro-6-(4-(1-(4-chloro-2-fluorobenzyl)piperidi...)
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50301351(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337235((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337220((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337217(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337211((S)-5-chloro-6-(4-(1-(2-chloro-4-fluorobenzyl)pipe...)
Affinity DataIC50: 58nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337261((S)-5-chloro-N-methyl-6-(3-methyl-4-(1-(trifluorom...)
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337223(5-chloro-6-(4-(1-(4-chlorobenzyl)-3-methylpiperidi...)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337231((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337232((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 83nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Mouse)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337217(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataIC50: 84nMAssay Description:Antagonist activity at mouse CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337260((S)-5-chloro-N-methyl-6-(3-methyl-4-(1-(4-methylbe...)
Affinity DataIC50: 87nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Rat)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337217(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataIC50: 97nMAssay Description:Antagonist activity at rat CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337245(methyl 4-(3-chloro-5-(methylcarbamoyl)pyridin-2-yl...)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337214((S)-5-chloro-6-(4-(1-(4-chlorobenzoyl)piperidin-4-...)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337221((3R)-4-(4-(4-(3,4-dimethylphenyl)but-1-en-2-yl)-2-...)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337243((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337229(5-chloro-6-(4-(4-(4-chlorobenzyl)piperazin-1-yl)-3...)
Affinity DataIC50: 280nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337230((S)-1-(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-...)
Affinity DataIC50: 520nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50301346(5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-yl)pi...)
Affinity DataIC50: 560nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337241((S)-azetidin-1-yl(5-chloro-6-(4-(1-(4-chlorobenzyl...)
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 3(Human)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50337244((S)-5-chloro-6-(4-(1-(4-chlorobenzyl)piperidin-4-y...)
Affinity DataIC50: 830nMAssay Description:Antagonist activity at human CXCR3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
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