Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50004497
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483424(CHEMBL1671951)
Affinity DataKd:  8.00E+5nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483425(CHEMBL1671952)
Affinity DataKd:  1.10E+6nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM1885(3-(5-bromopyridin-2-yl)-1-(2-phenylethyl)thiourea ...)
Affinity DataKd:  2.00E+3nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483426(CHEMBL1580138)
Affinity DataKd:  1.60E+6nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483427(CHEMBL1671953)
Affinity DataKd:  8.00E+5nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483428(CHEMBL1671954)
Affinity DataKd:  1.30E+6nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483429(CHEMBL1535399)
Affinity DataKd:  3.00E+4nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483430(CHEMBL1468531)
Affinity DataKd:  1.70E+6nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50356171(CHEMBL1087842)
Affinity DataKd:  7.00E+5nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50483431(PT-101 | CHEMBL316796)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to HIV1 reverse transcriptase by surface plasmon resonance based biosensor assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50478032(GW4511 | GW564511 | GW69564 | CHEMBL275658)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM50476133(CHEMBL373571 | VRX-480773)
Affinity DataIC50: 4nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed
TargetReverse transcriptase(Human immunodeficiency virus type 1)
Beactica

Curated by ChEMBL
LigandPNGBDBM1885(3-(5-bromopyridin-2-yl)-1-(2-phenylethyl)thiourea ...)
Affinity DataIC50: 15nMAssay Description:Inhibition of HIV1 reverse transcriptaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2020
Entry Details Article
PubMed