Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50035836
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 2.40nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 4.70nMAssay Description:Tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012950(CHEMBL330074 | 2-Hydroxy-3-[3-(1H-imidazol-4-yl)-2...)
Affinity DataIC50: 6.20nMAssay Description:Tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012950(CHEMBL330074 | 2-Hydroxy-3-[3-(1H-imidazol-4-yl)-2...)
Affinity DataIC50: 6.70nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetCathepsin D(Bovine)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 10nMAssay Description:Tested for inhibition of Cathepsin D from bovineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetPepsin A(Pig)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 18nMAssay Description:Tested for inhibition of pepsin from porcineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012952(CHEMBL330093 | 2-Hydroxy-3-[3-(1H-imidazol-4-yl)-2...)
Affinity DataIC50: 110nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012952(CHEMBL330093 | 2-Hydroxy-3-[3-(1H-imidazol-4-yl)-2...)
Affinity DataIC50: 270nMAssay Description:Tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228479(CHEMBL3349575)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50406108(CHEMBL2115235)
Affinity DataIC50: 2.10E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012949(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 2.30E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012949(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 2.50E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50406108(CHEMBL2115235)
Affinity DataIC50: 3.50E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50228479(CHEMBL3349575)
Affinity DataIC50: 4.20E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50406109(CHEMBL2114246)
Affinity DataIC50: 4.20E+3nMAssay Description:Tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50406109(CHEMBL2114246)
Affinity DataIC50: 4.20E+3nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetCathepsin D(Bovine)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 8.00E+4nMAssay Description:Tested for inhibition of Cathepsin D from bovineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetRenin(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 9.20E+4nMAssay Description:Tested for inhibition of renin from humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Rabbit)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for inhibition of Angiotensin I converting enzyme from rabbit.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetPepsin A(Pig)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for inhibition of pepsin from porcineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetChymotrypsin-C(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for inhibition of Chymotrypsinogen from bovineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetChymotrypsin-C(Human)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50012951(4-Cyclohexyl-2-hydroxy-3-[3-(1H-imidazol-4-yl)-2-(...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for inhibition of Chymotrypsinogen from bovineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Rabbit)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM912(PEPSTATIN | Pepstatine | N-[(3-Methyl-1-oxobutyl)-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Tested for inhibition of Angiotensin I converting enzyme from rabbit.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed