Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 50032698
LigandPNGBDBM15234(NSC221019 | Wortmannin, Wm | cid_312145 | CHEMBL42...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM15234(NSC221019 | Wortmannin, Wm | cid_312145 | CHEMBL42...)
Affinity DataIC50: 13nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM15234(NSC221019 | Wortmannin, Wm | cid_312145 | CHEMBL42...)
Affinity DataIC50: 15nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM15234(NSC221019 | Wortmannin, Wm | cid_312145 | CHEMBL42...)
Affinity DataIC50: 89nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333219(6-(6-methoxypyridin-3-yl)benzo[d]thiazol-2-amine |...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333220(5-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333220(5-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333215(7-morpholinoquinazolin-4(3H)-one | CHEMBL1645100)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333215(7-morpholinoquinazolin-4(3H)-one | CHEMBL1645100)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333222(3-(2-aminobenzo[d]thiazol-6-yl)phenol | CHEMBL1645...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333226(4-(5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl)-1...)
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333221(6-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333221(6-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333222(3-(2-aminobenzo[d]thiazol-6-yl)phenol | CHEMBL1645...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333221(6-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 9.70E+3nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333220(5-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333222(3-(2-aminobenzo[d]thiazol-6-yl)phenol | CHEMBL1645...)
Affinity DataIC50: 1.08E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333211(2-(pyridin-4-yl)thiazolo[5,4-d]pyrimidin-7-amine |...)
Affinity DataIC50: 1.11E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333216(4-(1H-pyrazolo[3,4-b]pyridin-4-yl)morpholine | CHE...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333222(3-(2-aminobenzo[d]thiazol-6-yl)phenol | CHEMBL1645...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333221(6-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333215(7-morpholinoquinazolin-4(3H)-one | CHEMBL1645100)
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333226(4-(5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl)-1...)
Affinity DataIC50: 1.42E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333210(5-(pyridin-4-yl)-1H-pyrrolo[2,3-b]pyridine | CHEMB...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333211(2-(pyridin-4-yl)thiazolo[5,4-d]pyrimidin-7-amine |...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333217(4-methyl-2-morpholinothiazole-5-carboxylic acid | ...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333216(4-(1H-pyrazolo[3,4-b]pyridin-4-yl)morpholine | CHE...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333217(4-methyl-2-morpholinothiazole-5-carboxylic acid | ...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50024966(6-Oxo-1,6-dihydro-[3,4']bipyridinyl-5-carbonitrile...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333211(2-(pyridin-4-yl)thiazolo[5,4-d]pyrimidin-7-amine |...)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50024966(6-Oxo-1,6-dihydro-[3,4']bipyridinyl-5-carbonitrile...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333217(4-methyl-2-morpholinothiazole-5-carboxylic acid | ...)
Affinity DataIC50: 2.76E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333216(4-(1H-pyrazolo[3,4-b]pyridin-4-yl)morpholine | CHE...)
Affinity DataIC50: 2.93E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333218(7-morpholinopyrimido[4,5-d]pyrimidin-4-amine | CHE...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333212(2-(pyridin-4-yl)benzo[d]oxazol-5-ol | CHEMBL164509...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333224(2-(dimethylamino)-6-morpholinopyrimidin-4(3H)-one ...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333218(7-morpholinopyrimido[4,5-d]pyrimidin-4-amine | CHE...)
Affinity DataIC50: 3.68E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333210(5-(pyridin-4-yl)-1H-pyrrolo[2,3-b]pyridine | CHEMB...)
Affinity DataIC50: 4.08E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333213(5-(pyridin-4-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-2...)
Affinity DataIC50: 4.30E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333218(7-morpholinopyrimido[4,5-d]pyrimidin-4-amine | CHE...)
Affinity DataIC50: 4.32E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333211(2-(pyridin-4-yl)thiazolo[5,4-d]pyrimidin-7-amine |...)
Affinity DataIC50: 4.35E+4nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333223(6-amino-2'-methyl-3,4'-bipyridine-5-carboxamide | ...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333213(5-(pyridin-4-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-2...)
Affinity DataIC50: 5.54E+4nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333225(1-methyl-1H-pyrrolo[2,3-c]pyridin-5-amine | CHEMBL...)
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333210(5-(pyridin-4-yl)-1H-pyrrolo[2,3-b]pyridine | CHEMB...)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of human p110alpha PI3K fragment by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333213(5-(pyridin-4-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-2...)
Affinity DataIC50: 6.20E+4nMAssay Description:Inhibition of human PI3K p110beta catalytic subunit by AlphaScreen competition assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50024966(6-Oxo-1,6-dihydro-[3,4']bipyridinyl-5-carbonitrile...)
Affinity DataIC50: 6.57E+4nMAssay Description:Inhibition of human PI3K p110delta catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333210(5-(pyridin-4-yl)-1H-pyrrolo[2,3-b]pyridine | CHEMB...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
LigandPNGBDBM50333220(5-(pyridin-4-yl)benzo[d]thiazol-2-amine | CHEMBL16...)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibition of human PI3K p110gamma catalytic subunit by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2011
Entry Details Article
PubMed
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