Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50039357
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335329(2-(4-Fluorobenzyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50: 14nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335315(2-(Methyl-3-pyridine)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 17nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335332(4-(1H-Pyrazol-3-ylamino)-2-p-tolyl-2H-phthalazin-1...)
Affinity DataIC50: 23nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335333(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-m-tolyl-2H-pht...)
Affinity DataIC50: 24nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249453(2-(2,5-difluorobenzyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 25nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335331(2-(4-Methoxyphenyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50: 29nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335330(4-(5-Methyl-2H-pyrazole-3-ylamino)phenyl-2H-phthal...)
Affinity DataIC50: 31nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335327(2-(4-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50: 32nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335323(2-Isopropyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-p...)
Affinity DataIC50: 35nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335322(2-(3-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50: 36nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335334(2-(4-Fluorophenyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50: 37nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335336(2-(3,5-Difluorobenzyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 49nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335324(2-(4-Toluylsulfonate)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 56nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335335(2-Benzyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-phth...)
Affinity DataIC50: 65nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249210(4-(5-methyl-1H-pyrazol-3-ylamino)-2-(2,2,2-trifluo...)
Affinity DataIC50: 66nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335337(2-[2-(4-Methoxyphenyl)-2-oxoethyl]-4-(5-methyl-1H-...)
Affinity DataIC50: 67nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249420(4-(5-methyl-1H-pyrazol-3-ylamino)-2-(2-oxo-2-pheny...)
Affinity DataIC50: 71nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249237(2-(4-chlorophenyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50: 93nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335317(N-{4-[1-Oxo-4-(1H-pyrazol-3-ylamino)-1H-phthalazin...)
Affinity DataIC50: 93nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335328(2-[2-(3-Methoxyphenyl)-2-oxoethyl]-4-(5-methyl-1H-...)
Affinity DataIC50: 100nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335340(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(4-nitrobenzyl...)
Affinity DataIC50: 109nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335325(2-Isobutyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-ph...)
Affinity DataIC50: 115nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335320(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(2-methylthiaz...)
Affinity DataIC50: 120nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335339(2-(4-tert-Butylphenyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 240nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335321(2-(Methyl-4-pyridine)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 270nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335318(2-Methyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-phth...)
Affinity DataIC50: 270nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335326(N-(4-((4-(1H-pyrazol-3-ylamino)-1-oxophthalazin-2(...)
Affinity DataIC50: 550nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335319(4-(5-Methyl-1H-pyrazol-3-ylamino)-2H-phthalazin-1-...)
Affinity DataIC50: 650nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335338(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-[2-oxo-2-(4-tr...)
Affinity DataIC50: 720nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335340(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(4-nitrobenzyl...)
Affinity DataIC50: 930nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335341(4-(1H-pyrazol-3-ylamino)-2-p-tolylphthalazin-1(2H)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335315(2-(Methyl-3-pyridine)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335316(4-(1H-Indazol-3-ylamino)-2-phenyl-2H-phthalazin-1-...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of Aurora A by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335317(N-{4-[1-Oxo-4-(1H-pyrazol-3-ylamino)-1H-phthalazin...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50249210(4-(5-methyl-1H-pyrazol-3-ylamino)-2-(2,2,2-trifluo...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335318(2-Methyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-phth...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335319(4-(5-Methyl-1H-pyrazol-3-ylamino)-2H-phthalazin-1-...)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335320(4-(5-Methyl-1H-pyrazol-3-ylamino)-2-(2-methylthiaz...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335321(2-(Methyl-4-pyridine)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335322(2-(3-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335323(2-Isopropyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-p...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335324(2-(4-Toluylsulfonate)-4-(5-methyl-1H-pyrazol-3-yla...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335325(2-Isobutyl-4-(5-methyl-1H-pyrazol-3-ylamino)-2H-ph...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335326(N-(4-((4-(1H-pyrazol-3-ylamino)-1-oxophthalazin-2(...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335327(2-(4-Methoxybenzyl)-4-(5-methyl-1H-pyrazol-3-ylami...)
Affinity DataIC50: 4.60E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335339(2-(4-tert-Butylphenyl)-4-(5-methyl-1H-pyrazol-3-yl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335328(2-[2-(3-Methoxyphenyl)-2-oxoethyl]-4-(5-methyl-1H-...)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335329(2-(4-Fluorobenzyl)-4-(5-methyl-1H-pyrazol-3-ylamin...)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335337(2-[2-(4-Methoxyphenyl)-2-oxoethyl]-4-(5-methyl-1H-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Evotec (Uk)

Curated by ChEMBL
LigandPNGBDBM50335332(4-(1H-Pyrazol-3-ylamino)-2-p-tolyl-2H-phthalazin-1...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of Aurora B by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/4/2013
Entry Details Article
PubMed
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