Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50033561
TargetHistone deacetylase 1(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 1(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 7nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 14nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 2(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant HDAC2 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 1(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC1 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase 6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 3(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 150nMAssay Description:Inhibition of human recombinant HDAC3 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 200nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 5(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HDAC5 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetHistone deacetylase 6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of human recombinant HDAC6 using fluor de Lys as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347387(CHEMBL1801172)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347387(CHEMBL1801172)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347387(CHEMBL1801172)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2C19(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347386(CHEMBL1801233)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2C19More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347386(CHEMBL1801233)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 2D6(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347385(CHEMBL1801250)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347386(CHEMBL1801233)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
Chroma Therapeutics

Curated by ChEMBL
LigandPNGBDBM50347384(CHEMBL1801238)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of CYP3A4More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed