Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50039318
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50367916(Metribolone | R-1881 | METHYLTRIENOLONE)
Affinity DataIC50: 7nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 10nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331713(5,7-dichloro-3-(trifluoromethyl)-1,2,3,4-tetrahydr...)
Affinity DataIC50: 13nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331698(5,6-dichloro-9H-carbazol-1-ol | CHEMBL1288959)
Affinity DataIC50: 15nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331708(6,7-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 27nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM8885(Testosterone, 1 | (1S,2R,10R,11S,14S,15S)-14-hydro...)
Affinity DataIC50: 30nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331697(2-bromo-6,7-dichloro-9H-carbazol-1-ol | CHEMBL1288...)
Affinity DataIC50: 34nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331710(6,7-dichloro-1-(perfluoroethyl)-2,3,4,9-tetrahydro...)
Affinity DataIC50: 34nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331701(6,8-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 34nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331702(5,8-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 85nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331704(8-chloro-6-fluoro-1-(trifluoromethyl)-2,3,4,9-tetr...)
Affinity DataIC50: 90nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331709(5,6-dichloro-1-(trifluoromethyl)-2,3,4,9-tetrahydr...)
Affinity DataIC50: 95nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331712(6,8-dichloro-2,2-difluoro-1-(trifluoromethyl)-2,3,...)
Affinity DataIC50: 100nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331707(1-hydroxy-1-(trifluoromethyl)-2,3,4,9-tetrahydro-1...)
Affinity DataIC50: 480nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331703(2,4-dichloro-6-(trifluoromethyl)-5,6,7,8,9,10-hexa...)
Affinity DataIC50: 600nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331700(2-benzyl-5,6-dichloro-9H-carbazol-1-ol | CHEMBL129...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331699(2-benzyl-6,7-dichloro-9H-carbazol-1-ol | CHEMBL129...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331695(6-bromo-9H-carbazol-1-ol | CHEMBL1288956)
Affinity DataIC50: 1.42E+3nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331696(8-hydroxy-9H-carbazole-3-carbonitrile | CHEMBL1288...)
Affinity DataIC50: 4.60E+3nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331706(1-hydroxy-1-methyl-2,3,4,9-tetrahydro-1H-carbazole...)
Affinity DataIC50: 9.20E+3nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331705(6,7-dichloro-1-methyl-2,3,4,9-tetrahydro-1H-carbaz...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetAndrogen receptor(Human)
Radius Health

Curated by ChEMBL
LigandPNGBDBM50331711(1-hydroxy-1-(perfluoroethyl)-2,3,4,9-tetrahydro-1H...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to androgen receptor by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed