Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50032487
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330034(Bis(3-bromophenyl)(4-hydroxy)thiosemicarbazone | C...)
Affinity DataIC50: 126nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330030([(3-Bromophenyl)-(3-hydroxyphenyl)-ketone]thiosemi...)
Affinity DataIC50: 131nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330031([(3-Bromophenyl)-(3-acetoxyphenyl)-ketone]thiosemi...)
Affinity DataIC50: 151nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330036(Bis(3-bromophenyl)(5-hydroxy)thiosemicarbazone | C...)
Affinity DataIC50: 232nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330041((3-Bromophenyl)(3-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 370nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330042((3-Bromophenyl)(4-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 815nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330043((3-Bromophenyl)(5-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 931nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330045((3-Bromobenzoylpyridine)thiosemicarbazone | CHEMBL...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330039([(3,4,5-Trimethoxyphenyl)-(4-methoxy,5-hydroxyphen...)
Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330031([(3-Bromophenyl)-(3-acetoxyphenyl)-ketone]thiosemi...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330039([(3,4,5-Trimethoxyphenyl)-(4-methoxy,5-hydroxyphen...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330051([2-Phenylacetophenone]thiosemicarbazone | CHEMBL12...)
Affinity DataIC50: 5.41E+3nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330034(Bis(3-bromophenyl)(4-hydroxy)thiosemicarbazone | C...)
Affinity DataIC50: 9.49E+3nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330049([(3-Bromophenyl)-(5,6,7,8-tetrahydronaphthalen-2-y...)
Affinity DataIC50: 9.65E+3nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330046(2-((3-bromophenyl)(6-bromopyridin-3-yl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330045((3-Bromobenzoylpyridine)thiosemicarbazone | CHEMBL...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330046(2-((3-bromophenyl)(6-bromopyridin-3-yl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330047(2-((3-bromophenyl)(2-bromopyridin-3-yl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330044([(3-Benzoylpyridine)-ketone]thiosemicarbazone | CH...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330049([(3-Bromophenyl)-(5,6,7,8-tetrahydronaphthalen-2-y...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330047(2-((3-bromophenyl)(2-bromopyridin-3-yl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330048([(3-Bromophenyl)-cyclohexylketone]thiosemicarbazon...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330048([(3-Bromophenyl)-cyclohexylketone]thiosemicarbazon...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330041((3-Bromophenyl)(3-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330050([Bis-diphenylketone]thiosemicarbazone | CHEMBL1269...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330050([Bis-diphenylketone]thiosemicarbazone | CHEMBL1269...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330051([2-Phenylacetophenone]thiosemicarbazone | CHEMBL12...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330052([9-Fluorenone]-thiosemicarbazone | CHEMBL1269811)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330052([9-Fluorenone]-thiosemicarbazone | CHEMBL1269811)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330053([2,7-Dibromo-9H-fluoren-9-one]-thiosemicarbazone |...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330053([2,7-Dibromo-9H-fluoren-9-one]-thiosemicarbazone |...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330037([5-Bromo(t-butyldimethylsilyl)oxyphenyl-]-(3-bromo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330029((3-Hydroxyphenyl)thiosemicarbazone | CHEMBL1269631)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330030([(3-Bromophenyl)-(3-hydroxyphenyl)-ketone]thiosemi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330032(2-((3-(benzyloxy)phenyl)(3-bromophenyl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330032(2-((3-(benzyloxy)phenyl)(3-bromophenyl)methylene)h...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330033([[3-(t-Butyldimethylsilyl)oxyphenyl]-(3-bromopheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330033([[3-(t-Butyldimethylsilyl)oxyphenyl]-(3-bromopheny...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330035([4-Bromo(t-butyldimethylsilyl)oxyphenyl-]-(3-bromo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330035([4-Bromo(t-butyldimethylsilyl)oxyphenyl-]-(3-bromo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330036(Bis(3-bromophenyl)(5-hydroxy)thiosemicarbazone | C...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330044([(3-Benzoylpyridine)-ketone]thiosemicarbazone | CH...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330037([5-Bromo(t-butyldimethylsilyl)oxyphenyl-]-(3-bromo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330038(2-((3-bromo-2-hydroxyphenyl)(3-bromophenyl)methyle...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330038(2-((3-bromo-2-hydroxyphenyl)(3-bromophenyl)methyle...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330040([(3-Benzoylthiophene)-ketone]thiosemicarbazone | C...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330040([(3-Benzoylthiophene)-ketone]thiosemicarbazone | C...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetProcathepsin L(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330029((3-Hydroxyphenyl)thiosemicarbazone | CHEMBL1269631)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin L after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330042((3-Bromophenyl)(4-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
TargetCathepsin B(Human)
Baylor University

Curated by ChEMBL
LigandPNGBDBM50330043((3-Bromophenyl)(5-bromothiophene)thiosemicarbazone...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human liver cathepsin B after 5 mins by microplate reader analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed