Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 5041
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84968(Urea derivative, 12)
Affinity DataKi:  3.20E+3nM IC50: 8.40E+3nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84969(Urea derivative, 13)
Affinity DataKi:  4.60E+3nM IC50: 1.43E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84967(Urea derivative, 11)
Affinity DataKi:  7.20E+3nM IC50: 1.98E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84972(Urea derivative, 16)
Affinity DataKi:  9.40E+3nM IC50: 1.85E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84963(Urea derivative, 7)
Affinity DataKi:  1.05E+4nM IC50: 1.95E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84962(Urea derivative, 6)
Affinity DataKi:  1.06E+4nM IC50: 4.21E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84966(Urea derivative, 10)
Affinity DataKi:  1.21E+4nM IC50: 2.88E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84970(Urea derivative, 14)
Affinity DataKi:  1.70E+4nM IC50: 2.91E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM18351((2R,3R,4R,5S)-2-(hydroxymethyl)piperidine-3,4,5-tr...)
Affinity DataKi:  1.80E+4nM IC50: 3.95E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataKi:  2.15E+4nM IC50: 2.64E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84959(Stilbene derivative, 2)
Affinity DataKi:  3.51E+4nM IC50: 4.64E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84973(Urea derivative, 17)
Affinity DataIC50: 5.88E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84971(Urea derivative, 15)
Affinity DataIC50: 6.01E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84965(Urea derivative, 9)
Affinity DataIC50: 6.36E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84975(Urea derivative, 19)
Affinity DataIC50: 6.43E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84964(Urea derivative, 8)
Affinity DataIC50: 6.85E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM50322066(CHEMBL1172402 | Stilbene derivative, 3 | 3,5-Dihyd...)
Affinity DataIC50: 1.02E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84974(Urea derivative, 18)
Affinity DataIC50: 1.05E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84961(Stilbene derivative, 5)
Affinity DataIC50: 2.00E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM84960(Stilbene derivative, 4)
Affinity DataIC50: 2.00E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Gyeongsang National University

LigandPNGBDBM50173649(CHEMBL194754 | Stilbene derivative, 1 | 4-[(E)-2-(...)
Affinity DataIC50: 2.00E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2012
Entry Details Article
PubMed