Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50032366
TargetSecretin receptor(Human)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327887(HSDGTFTSELSRLQDSARLQRLLQGLV-NH2 | CHEMBL1255581)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at secretin receptor expressed in CHO cells assessed as increase of cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSecretin receptor(Human)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327888(CHEMBL1256314)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at secretin receptor expressed in CHO cells assessed as increase of cAMP levelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSecretin receptor(Human)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327887(HSDGTFTSELSRLQDSARLQRLLQGLV-NH2 | CHEMBL1255581)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]-secretin-27 from secretin receptor expressed in CHO cells by gamma-spectrometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed
TargetSecretin receptor(Human)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50327888(CHEMBL1256314)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]-secretin-27 from secretin receptor expressed in CHO cells by gamma-spectrometer analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/12/2011
Entry Details Article
PubMed