Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 50001068
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 0.600nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012313(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012306(CHEMBL274874 | Ac-His-Trp-Ala-Val-Gly-His-Leu-Met-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012311(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012307(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012308(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 3nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012309(CHEMBL263873 | Ac-His-Trp-Ala-Val-D-Ala-His-Leu-Me...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012297(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012300(2-[2-[2-(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 4nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012314(CHEMBL440986 | (CH3)CCO-His-Trp-Ala-Val-Gly-His-Le...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012312(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012319(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 5nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012311(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 6nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012301(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 6.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012308(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 7nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012313(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 8nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012307(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 10nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012303(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 11nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012297(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 11nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012310(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 18nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012315(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 18nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012310(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 18nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012300(2-[2-[2-(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 20nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012303(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 22nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012301(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 31nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012316(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 32nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012316(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 32nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012312(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 35nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012319(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 35nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012315(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 80nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012299(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 81nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012302(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 91nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012302(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 91nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012298(CHEMBL438290 | Ac-His-Trp-Ala-Val-Ala-His-Leu-Met-...)
Affinity DataIC50: 180nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012305(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 300nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012299(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 300nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50012305(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 410nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed