Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50001064
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012292(CHEMBL414570 | AcMet-Val-Val-Ala-Ser-Gln-Leu-Arg-A...)
Affinity DataKi:  5.00E+4nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012291(CHEMBL429238 | Phe-Thr-Glu-Met-Met-Val-Val-Ala-Ser...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012296(CHEMBL413040 | Ac-Ile-Ser-His-Lys-Asp-Met-Gln-Leu-...)
Affinity DataKi:  1.00E+5nMAssay Description:Compound was tested for the inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor binding to PMNL membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012294(CHEMBL438915 | AcMet-Ile-Lys-Ala-Phe-Thr-Glu-Met-M...)
Affinity DataKi:  1.00E+5nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012290(2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(3H-imidazol-...)
Affinity DataKi:  1.50E+5nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012293(CHEMBL409278 | Ser-Gln-Leu-Alr-Ala-Asn-Ile-Ser-His...)
Affinity DataKi:  3.00E+5nMAssay Description:Compound was tested for the inhibition of [125I]C5a anaphylatoxin chemotactic receptor binding to PMNL membranes at a concentration of 0.1-1 mMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50012295(Ile-Ser-His-Lys-Asp-Met-Gln-Leu-Gly-Arg | CHEMBL21...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC5a anaphylatoxin chemotactic receptor 1(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50008376(2-[2-(2-{2-[2-(2-{6-Amino-2-[2-amino-3-(3H-imidazo...)
Affinity DataKi:  3.00E+5nMAssay Description:Inhibition of [125I]C5a binding to C5a anaphylatoxin chemotactic receptor in PMNL membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed