Compile Data Set for Download or QSAR
Report error Found 56 Enz. Inhib. hit(s) with all data for entry = 5782
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93422(PHD Inhibitor, 12{1,1,2})
Affinity DataIC50: 4.30nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93422(PHD Inhibitor, 12{1,1,2})
Affinity DataIC50: 4.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93425(PHD Inhibitor, 12{4,1,2})
Affinity DataIC50: 5.10nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 5.30nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93430(PHD Inhibitor, 12{2,1,2})
Affinity DataIC50: 6.40nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 7.20nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93426(PHD Inhibitor, 12{2,5,2})
Affinity DataIC50: 7.60nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 8.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93426(PHD Inhibitor, 12{2,5,2})
Affinity DataIC50: 8.90nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93427(PHD Inhibitor, 12{2,6,2})
Affinity DataIC50: 11nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 11.7nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 12.2nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 12.6nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 12.9nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 13.2nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93425(PHD Inhibitor, 12{4,1,2})
Affinity DataIC50: 13.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 13.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93430(PHD Inhibitor, 12{2,1,2})
Affinity DataIC50: 13.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93432(PHD Inhibitor, 12{2,6,4})
Affinity DataIC50: 14.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 14.6nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93427(PHD Inhibitor, 12{2,6,2})
Affinity DataIC50: 16.2nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93432(PHD Inhibitor, 12{2,6,4})
Affinity DataIC50: 16.8nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93433(PHD Inhibitor, 12{2,1,4})
Affinity DataIC50: 18.8nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 20nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 22nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93420(PHD Inhibitor, 12{3,1,4})
Affinity DataIC50: 32nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93422(PHD Inhibitor, 12{1,1,2})
Affinity DataIC50: 35nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 37.4nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93419(PHD Inhibitor, 12{2,4,1})
Affinity DataIC50: 38.3nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93418(PHD Inhibitor, 12{2,3,1})
Affinity DataIC50: 40nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93425(PHD Inhibitor, 12{4,1,2})
Affinity DataIC50: 41.9nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93426(PHD Inhibitor, 12{2,5,2})
Affinity DataIC50: 44.8nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93418(PHD Inhibitor, 12{2,3,1})
Affinity DataIC50: 49nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93433(PHD Inhibitor, 12{2,1,4})
Affinity DataIC50: 60.8nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93427(PHD Inhibitor, 12{2,6,2})
Affinity DataIC50: 67.5nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93420(PHD Inhibitor, 12{3,1,4})
Affinity DataIC50: 77nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 86.4nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93423(PHD Inhibitor, 12{2,3,2} | PHD Inhibitor, 12{2,4,2...)
Affinity DataIC50: 90.2nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93430(PHD Inhibitor, 12{2,1,2})
Affinity DataIC50: 93.8nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN2(Human)
Amgen

LigandPNGBDBM93421(PHD Inhibitor, 12{1,5,3})
Affinity DataIC50: 95nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93428(PHD Inhibitor, 12{2,3,4} | PHD Inhibitor, 12{2,4,4...)
Affinity DataIC50: 104nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93412(PHD Inhibitor, 8{2})
Affinity DataIC50: 112nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93432(PHD Inhibitor, 12{2,6,4})
Affinity DataIC50: 113nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93416(PHD Inhibitor, 8{6})
Affinity DataIC50: 138nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetProlyl hydroxylase EGLN3(Human)
Amgen

LigandPNGBDBM93421(PHD Inhibitor, 12{1,5,3})
Affinity DataIC50: 165nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93415(PHD Inhibitor, 8{5})
Affinity DataIC50: 265nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93414(PHD Inhibitor, 8{4})
Affinity DataIC50: 293nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93433(PHD Inhibitor, 12{2,1,4})
Affinity DataIC50: 308nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93417(PHD Inhibitor, 8{7})
Affinity DataIC50: 409nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
TargetEgl nine homolog 1(Human)
Amgen

LigandPNGBDBM93411(PHD Inhibitor, 8{1})
Affinity DataIC50: 482nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/17/2013
Entry Details Article
PubMed
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