Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50032146
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324887(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-n...)
Affinity DataKi:  1.69nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324887(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-n...)
Affinity DataKi:  2.32nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  2.75nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324894(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)naph...)
Affinity DataKi:  2.87nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324890(N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)naph...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324889(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2-...)
Affinity DataKi:  4.59nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50261126(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)nap...)
Affinity DataKi:  4.64nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324888(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)naph...)
Affinity DataKi:  5.19nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324893(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)-2-n...)
Affinity DataKi:  6.15nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324892(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)nap...)
Affinity DataKi:  8.53nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324891(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-2-...)
Affinity DataKi:  9.36nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324894(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)naph...)
Affinity DataKi:  9.62nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324891(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-2-...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [3H]MK912 from human alpha2A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324889(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2-...)
Affinity DataKi:  17.8nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  20.2nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324888(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)naph...)
Affinity DataKi:  24.4nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324892(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)nap...)
Affinity DataKi:  27.4nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324890(N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)naph...)
Affinity DataKi:  46.5nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324891(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-2-...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324890(N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)naph...)
Affinity DataKi:  62nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324889(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)-2-...)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324890(N-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)naph...)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324892(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)nap...)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324893(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)-2-n...)
Affinity DataKi:  96nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324894(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)naph...)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50261126(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)nap...)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324893(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)-2-n...)
Affinity DataKi:  102nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50261126(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)nap...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324887(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-n...)
Affinity DataKi:  113nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324893(N-(6-(4-(2-methoxyphenyl)piperazin-1-yl)hexyl)-2-n...)
Affinity DataKi:  121nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50261126(N-(3-(4-(2-methoxyphenyl)piperazin-1-yl)propyl)nap...)
Affinity DataKi:  132nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50119380(CHEMBL540612 | N-(4-(4-(2-methoxyphenyl)piperazin-...)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]8OH-DPAT from human 5HT1A receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324891(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)-2-...)
Affinity DataKi:  254nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324888(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)naph...)
Affinity DataKi:  348nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324892(N-(5-(4-(2-methoxyphenyl)piperazin-1-yl)pentyl)nap...)
Affinity DataKi:  438nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of LièGe

Curated by ChEMBL
LigandPNGBDBM50324887(N-(2-(4-(2-methoxyphenyl)piperazin-1-yl)ethyl)-2-n...)
Affinity DataKi:  890nMAssay Description:Displacement of [3H]spiperone from human D2L receptor after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/20/2011
Entry Details Article
PubMed